SCHEMBL20754196

SCHEMBL20754196

CCn1nncc1C(C)C

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 1/20 0.33
SLC9A1 P19634 1/20 0.31
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25744948 0.83 TOP2A (0.36) TOP2ASLC9A1
SCHEMBL18460627 0.83 NPC1 (0.35) TOP2APTGS2
SCHEMBL18460735 0.83 NPC1 (0.35) TOP2APTGS2
SCHEMBL24665883 0.81 TOP2A (0.32) TOP2A
SCHEMBL20711389 0.81 TOP2A (0.39) TOP2A
SCHEMBL25857817 0.80 TOP2A (0.39) TOP2ASLC9A1
SCHEMBL25744939 0.78
SCHEMBL19303015 0.77 NPC1 (0.32)
SCHEMBL24769809 0.75
SCHEMBL24380279 0.75 KMT2A (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12024507-B2 Compounds as GLP-1R agonists TERNS PHARMACEUTICALS, INC. (US) 2024-07-02 US disclosed
US-20230357254-A1 IMIDAZOPYRIDAZINES AS MODULATORS OF IL-17 JANSSEN PHARMACEUTICA NV (BE) 2023-11-09 US disclosed
US-20230357254-A1 IMIDAZOPYRIDAZINES AS MODULATORS OF IL-17 JANSSEN PHARMACEUTICA NV (BE) 2023-11-09 US disclosed
US-11746113-B2 Labelled cannabinergic ligands and related analogs MAKRIYANNIS ALEXANDROS (US) 2023-09-05 US disclosed
US-11702422-B2 Imidazopyridazines as modulators of IL-17 JANSSEN PHARMACEUTICA NV (BE) 2023-07-18 US disclosed
US-11702422-B2 Imidazopyridazines as modulators of IL-17 JANSSEN PHARMACEUTICA NV (BE) 2023-07-18 US disclosed
US-11691979-B2 Imidazopyridazines as modulators of IL-17 JANSSEN PHARMACEUTICA NV (BE) 2023-07-04 US disclosed
US-11691979-B2 Imidazopyridazines as modulators of IL-17 JANSSEN PHARMACEUTICA NV (BE) 2023-07-04 US disclosed
US-20230159512-A1 COMPOUNDS AS GLP-1R AGONISTS TERNS PHARMACEUTICALS, INC. 2023-05-25 US disclosed
US-20230159512-A1 COMPOUNDS AS GLP-1R AGONISTS TERNS PHARMACEUTICALS, INC. 2023-05-25 US disclosed
US-11247990-B1 Bicyclic fused pyridine compounds as inhibitors of TAM kinases ARRAY BIOPHARMA INC (US) 2022-02-15 US disclosed
US-11174281-B1 Modified nucleotides and uses thereof Singular Genomics Systems, Inc. (US) 2021-11-16 US disclosed
US-20210316006-A1 PYRROLOBENZODIAZEPINE CONJUGATES MEDIMMUNE LIMITED (GB) 2021-10-14 US disclosed
US-20210300937-A1 Novel Labelled Cannabinergic Ligands and Related Analogs MAKRIYANNIS ALEXANDROS (US) 2021-09-30 US disclosed
US-20200361980-A1 14-MEMBERED KETOLIDES AND METHODS OF THEIR PREPARATION AND USE PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2020-11-19 US disclosed
US-20200306243-A1 COMPOUNDS AND CONJUGATES THEREOF MEDIMMUNE LIMITED (GB) 2020-10-01 US disclosed
US-RE48175-E1 Hydrophobically tagged small molecules as inducers of protein degradation DANA-FARBER CANCER INSTITUTE, INC. (US) 2020-08-25 US disclosed
US-20190330157-A1 THERAPEUTIC COMPOUNDS REGENTS OF THE UNIVERSITY OF MINNESOTA 2019-10-31 US disclosed
US-10392393-B2 Pyrrolobenzodiazepines MEDIMMUNE LIMITED (GB) 2019-08-27 US disclosed
US-20190055254-A1 PYRROLOBENZODIAZEPINES MEDIMMUNE LIMITED (GB) 2019-02-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (15 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11691979-B2 Imidazopyridazines as modulators of IL-17 IL17A, IL23R, IL15 TOP2A 2735/4885SLC9A1 3879/4885PTGS2 491/4885
US-20230357254-A1 IMIDAZOPYRIDAZINES AS MODULATORS OF IL-17 IL17A, IL23R, IL15 TOP2A 2735/4885SLC9A1 3879/4885PTGS2 491/4885
US-20190330157-A1 THERAPEUTIC COMPOUNDS OPRL1, INA, OGFR TOP2A 4182/4885SLC9A1 1003/4885PTGS2 1337/4885
US-11746113-B2 Labelled cannabinergic ligands and related analogs CNR1, CNR2, CHRND TOP2A 4395/4885SLC9A1 1564/4885PTGS2 1146/4885
US-12024507-B2 Compounds as GLP-1R agonists GLP1R, GIPR, GCGR TOP2A 4794/4885SLC9A1 378/4885PTGS2 2778/4885
US-20190055254-A1 PYRROLOBENZODIAZEPINES HRH3, HRH4, HRH2 TOP2A 953/4885SLC9A1 2297/4885PTGS2 1244/4885
US-20230159512-A1 COMPOUNDS AS GLP-1R AGONISTS GLP1R, GIPR, GCGR TOP2A 4815/4885SLC9A1 409/4885PTGS2 2777/4885
US-20200306243-A1 COMPOUNDS AND CONJUGATES THEREOF TOP2A, TOP1, TOP2B TOP2A 1/4885SLC9A1 4426/4885PTGS2 3636/4885
US-11702422-B2 Imidazopyridazines as modulators of IL-17 IL17A, IL23R, IL15 TOP2A 2735/4885SLC9A1 3879/4885PTGS2 491/4885
US-20210316006-A1 PYRROLOBENZODIAZEPINE CONJUGATES BCR, MCL1, CD79B TOP2A 50/4885SLC9A1 3023/4885PTGS2 4625/4885
US-11174281-B1 Modified nucleotides and uses thereof NUDT1, RNMT, ADAR TOP2A 623/4885SLC9A1 2987/4885PTGS2 2718/4885
US-11247990-B1 Bicyclic fused pyridine compounds as inhibitors of TAM kinases MAP3K1, MAP3K3, MAP3K2 TOP2A 2719/4885SLC9A1 3877/4885PTGS2 2313/4885
US-20210300937-A1 Novel Labelled Cannabinergic Ligands and Related Analogs CNR1, CNR2, CHRND TOP2A 4463/4885SLC9A1 1532/4885PTGS2 1188/4885
US-10392393-B2 Pyrrolobenzodiazepines HRH3, HRH4, HRH2 TOP2A 953/4885SLC9A1 2297/4885PTGS2 1244/4885
US-20200361980-A1 14-MEMBERED KETOLIDES AND METHODS OF THEIR PREPARATION AND USE CYP51A1, KHK, HSD17B7 TOP2A 1360/4885SLC9A1 4765/4885PTGS2 642/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.