SCHEMBL20846010

SCHEMBL20846010

COCCC(=O)N(C(=O)CCOC)c1ncc(-c2cncc(F)c2)nc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 9/20 0.35
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
KDR P35968 1/20 0.33
PTGES O14684 2/20 0.32
TLR7 Q9NYK1 3/20 0.31
DYRK1A Q13627 1/20 0.31
WNT1 P04628 1/20 0.30
CYP3A4 P08684 1/20 0.30
ADORA2A P29274 1/20 0.30
ADORA1 P30542 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20845987 0.86 ABL1 (0.35) ABL1PTGESTLR7DYRK1A
SCHEMBL20839264 0.82 CYP11B2 (0.36) ABL1PTGESDYRK1A
SCHEMBL20843729 0.80 ABL1 (0.33) ABL1PTGESTLR7DYRK1AADORA2A
SCHEMBL24013175 0.74 PTGES (0.33) ABL1PTGESTLR7
SCHEMBL19406218 0.73 KDR (0.42) ABL1HCRTR1HCRTR2KDRPTGES
SCHEMBL19406423 0.73 SMN1; SMN2 (0.35) ABL1HCRTR1HCRTR2PTGESTLR7
SCHEMBL20846004 0.72 KDM4E (0.34) ABL1
SCHEMBL19406487 0.71 TLR7 (0.34) ABL1HCRTR1HCRTR2PTGESTLR7
SCHEMBL20846007 0.69 KDR (0.43) HCRTR1HCRTR2KDRDYRK1ACYP3A4
SCHEMBL20845492 0.69 ABL1 (0.38) ABL1KDRDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11678665-B2 Pyrazine-4-carbamate or -urea derivatives as herbicides SYNGENTA PARTICIPATIONS AG (CH) 2023-06-20 US disclosed
US-11678665-B2 Pyrazine-4-carbamate or -urea derivatives as herbicides SYNGENTA PARTICIPATIONS AG (CH) 2023-06-20 US disclosed
EP-3684764-B1 PYRAZINE-4-CARBAMATE DERIVATIVES AS HERBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2021-11-10 EP disclosed
US-20200267983-A1 Pyrazine-4Carbamate or -Urea Derivatives As Herbicides SYNGENTA PARTICIPATIONS AG (CH) 2020-08-27 US disclosed
WO-2019057724-A1 PYRAZINE-4CARBAMATE OR -UREA DERIVATIVES AS HERBICIDES SYNGENTA PARTICIPATIONS AG (CH) 2019-03-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11678665-B2 Pyrazine-4-carbamate or -urea derivatives as herbicides DDT, PLPBP, CPS1 ABL1 2259/4885HCRTR1 2739/4885HCRTR2 3417/4885
US-20200267983-A1 Pyrazine-4Carbamate or -Urea Derivatives As Herbicides PLPBP, PDXK, HPD ABL1 2740/4885HCRTR1 2735/4885HCRTR2 3309/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.