SCHEMBL20899861

SCHEMBL20899861

CN(C(=O)Cc1cscn1)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLQ O75417 5/20 0.46
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
OPRD1 P41143 1/20 0.42
PKM P14618 1/20 0.42
LMNA P02545 1/20 0.41
TP53 P04637 1/20 0.41
MAPT P10636 1/20 0.41
GAA P10253 1/20 0.41
HPGD P15428 1/20 0.41
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
SLC6A3 Q01959 1/20 0.40
MAPK1 P28482 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7275089 0.78 MAPK1 (0.41) KMT2AMEN1OPRD1PKMLMNA
SCHEMBL5693351 0.75 MAPK1 (0.43) KMT2AMEN1OPRD1PKMLMNA
SCHEMBL7094417 0.73 MAPK1 (0.44) KMT2AMEN1OPRD1PKMLMNA
SCHEMBL8263373 0.72 ALDH1A1 (0.58) POLQKMT2AMEN1LMNAROCK2
SCHEMBL20899886 0.72 MAPK1 (0.47) KMT2AMEN1OPRD1PKMLMNA
SCHEMBL5071504 0.72 LMNA (0.48) POLQKMT2AMEN1PKMLMNA
SCHEMBL11438169 0.72 ROCK2 (0.47) POLQKMT2AMEN1LMNATP53
SCHEMBL20346360 0.70 POLQ (0.49) POLQKMT2AMEN1LMNATP53
SCHEMBL1760632 0.69 KMT2A (0.58) POLQKMT2AMEN1LMNANPSR1
SCHEMBL7830345 0.68 KMT2A (0.56) POLQKMT2AMEN1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019075394-A1 COMPOUNDS FOR TREATMENT OF EMOTIONAL/PSYCHOLOGICAL SYMPTOMS IN FRAGILE X SYNDROME VANDERKLISH PETER (US) 2019-04-18 WO disclosed