Cianopramine

Cianopramine

SCHEMBL209730

CN(C)CCCN1c2ccccc2CCc2ccc(C#N)cc21

nearest known ligand 0.78

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 16/20 0.78
LMNA P02545 3/20 0.71
MAPT P10636 3/20 0.71
HRH1 P35367 3/20 0.71
SLC22A1 O15245 2/20 0.71
CHRM2 P08172 2/20 0.71
CHRM4 P08173 2/20 0.71
HTR1A P08908 2/20 0.71
CHRM5 P08912 2/20 0.71
ADORA3 P0DMS8 2/20 0.71
CYP2D6 P10635 2/20 0.71
CHRM1 P11229 2/20 0.71
DRD2 P14416 2/20 0.71
ADRA2B P18089 2/20 0.71
ADRA2C P18825 2/20 0.71
CHRM3 P20309 2/20 0.71
DRD1 P21728 2/20 0.71
SLC6A2 P23975 2/20 0.71
HRH2 P25021 2/20 0.71
HTR2A P28223 2/20 0.71

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Imipramine SCHEMBL15719828 0.84 LMNA (0.97) SLC6A4LMNAMAPTHRH1SLC22A1
Imipramine SCHEMBL6118138 0.84 SLC6A4 (1.00) SLC6A4LMNAMAPTHRH1SLC22A1
Imipramine SCHEMBL29350100 0.84 SLC6A4 (1.00) SLC6A4LMNAMAPTHRH1SLC22A1
Imipramine SCHEMBL17004048 0.84 SLC6A4 (1.00) SLC6A4LMNAMAPTHRH1SLC22A1
Imipramine SCHEMBL34282 0.84 SLC6A4 (1.00) SLC6A4LMNAMAPTHRH1SLC22A1
SCHEMBL14732502 0.84 SLC6A4 (0.57) SLC6A4LMNAMAPTHRH1SLC22A1
SCHEMBL14723083 0.83 SLC6A4 (0.55) SLC6A4LMNAMAPTHRH1SLC22A1
SCHEMBL14723391 0.83 SLC6A4 (0.55) SLC6A4LMNAMAPTHRH1SLC22A1
Imipramine SCHEMBL41765 0.83 LMNA (1.00) SLC6A4LMNAMAPTHRH1SLC22A1
Imipramine SCHEMBL28759733 0.83 LMNA (1.00) SLC6A4LMNAMAPTHRH1SLC22A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 726 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240307393-A1 PHARMACEUTICAL COMPOSITION FOR CANCER PREVENTION OR TREATMENT, COMPRISING CDK4/6 INHIBITOR AND TRICYCLIC ANTIDEPRESSANT NATIONAL CANCER CENTER (KR) 2024-09-19 US claimed
EP-4368183-A1 PHARMACEUTICAL COMPOSITION FOR CANCER PREVENTION OR TREATMENT, COMPRISING CDK4/6 INHIBITOR AND TRICYCLIC ANTIDEPRESSANT National Cancer Center (KR) 2024-05-15 EP claimed
WO-2023282544-A1 PHARMACEUTICAL COMPOSITION FOR CANCER PREVENTION OR TREATMENT, COMPRISING CDK4/6 INHIBITOR AND TRICYCLIC ANTIDEPRESSANT 국립암센터 2023-01-12 WO claimed
WO-2022159506-A1 DEUTERATED CANNABIDIOL COMPOUNDS MERIT THERAPEUTICS, INC. (US) 2022-07-28 WO claimed
WO-2022159507-A1 COMBINATION OF CANNABINOIDS WITH ADDITIONAL THERAPEUTIC AGENTS FOR TREATING DISEASES OR DISORDERS MERIT THERAPEUTICS, INC. (US) 2022-07-28 WO claimed
US-20160303103-A1 COMPOUNDS THAT TREAT MALARIA AND PREVENT MALARIA TRANSMISSION THE USA, AS REPRESENTED BY THE SECRETARY, DEPT. OF HEALTH AND HUMAN SERVICES 2016-10-20 US claimed
CN-105636438-A Pharmaceutical composition comprising an AMPK activator and a serotonin active agent and uses thereof CHEN JIANHONG 2016-06-01 CN claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-20140350064-A1 PHARMACEUTICAL COMPOSITION COMPRISING AN AMPK ACTIVATOR AND A SEROTONERGIC AGENT AND METHODS OF USE THEREOF ALS MOUNTAIN LLC 2014-11-27 US claimed
CN-102143961-B Benzoxazines, benzothiazines, and related compounds having NOS inhibitory activity NEURAXON INC 2014-11-05 CN claimed
US-20010008896-A1 Administration of active agents, including 5-HT receptor agonists and antagonists, to treat premature ejaculation SMITH WILLIAM L (US) 2001-07-19 US claimed
EP-1096927-A1 COMPOSITION FOR TREATMENT OF STRESS Massachusetts Institute of Technology (US) 2001-05-09 EP claimed
WO-2000003701-A1 COMPOSITION FOR TREATMENT OF STRESS MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2000-01-27 WO claimed
US-5922341-A Local administration of pharmacologically active agents to treat premature ejaculation VIVUS, INCORPORATED (US) 1999-07-13 US claimed
EP-0386117-B1 TREATING PREMENSTRUAL OR LATE LUTEAL PHASE SYNDROME MASSACHUSETTS INST TECHNOLOGY (US) 1999-01-07 EP claimed
WO-1992000103-A1 PHARMACEUTICAL PREPARATIONS BEECHAM GROUP PLC (GB) 1992-01-09 WO claimed
EP-0440704-A1 COMPOSITIONS FOR TREATING TOBACCO WITHDRAWEL SYMPTOMS. MASSACHUSETTS INST TECHNOLOGY (US) 1991-08-14 EP claimed
EP-0386117-A1 TREATING PREMENSTRUAL OR LATE LUTEAL PHASE SYNDROME MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1990-09-12 EP claimed
WO-1990004387-A2 COMPOSITIONS FOR TREATING TOBACCO WITHDRAWAL SYMPTOMS MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1990-05-03 WO claimed
WO-1989003692-A1 TREATING PREMENSTRUAL OR LATE LUTEAL PHASE SYNDROME MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 1989-05-05 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160303103-A1 COMPOUNDS THAT TREAT MALARIA AND PREVENT MALARIA TRANSMISSION ICMT, MAVS, G6PD SLC6A4 3685/4885LMNA 2419/4885MAPT 520/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.