SCHEMBL2104832

SCHEMBL2104832

N#Cc1ccc2c(c1)=COCN=2

nearest known ligand 0.33

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.33
MAOB P27338 1/20 0.31
DRD2 P14416 2/20 0.31
DRD3 P35462 2/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
PNMT P11086 1/20 0.31
VCAM1 P19320 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19926284 0.61 CYP2A6 (0.37) CYP2A6DRD2DRD3CA1CA2
SCHEMBL1435831 0.61 ALDH1A1 (0.39) CYP2A6DRD2DRD3CA1CA2
SCHEMBL20204992 0.61 CA2 (0.40) CYP2A6CA1CA2VCAM1
SCHEMBL28971640 0.58 TSHR (0.63) CYP2A6MAOBDRD2DRD3CA2
SCHEMBL6739755 0.58
SCHEMBL15619538 0.58 IMPDH2 (0.32) MAOBDRD2DRD3CA1CA2
SCHEMBL9289 0.57 TSHR (0.61) DRD2DRD3
Water SCHEMBL28137572 0.57 TSHR (0.61) DRD2DRD3
SCHEMBL2817154 0.57 TSHR (0.61) DRD2DRD3
Bromide SCHEMBL17202846 0.57 PNMT (0.52) CYP2A6DRD2DRD3CA2PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116670115-A Process for preparing anthranilic acid/anthranilic acid amide compounds and intermediates thereof 皮埃企业有限公司 2023-08-29 CN disclosed
US-8163740-B2 6-substituted benzoxazines HOFFMANN-LA ROCHE INC. (US) 2012-04-24 US disclosed
US-20100063037-A1 6-SUBSTITUTED BENZOXAZINES F. HOFFMANN-LA ROCHE AG (CH) 2010-03-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100063037-A1 6-SUBSTITUTED BENZOXAZINES HTR5A, NPY5R, GABRA5 CYP2A6 379/4885MAOB 161/4885DRD2 71/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.