SCHEMBL21048813

SCHEMBL21048813

CCS(=O)(=O)N(C)c1ccccc1CNC(=O)O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.41
GAA P10253 1/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 4/20 0.41
HPGD P15428 2/20 0.41
JAK2 O60674 4/20 0.41
JAK1 P23458 4/20 0.41
TYK2 P29597 4/20 0.41
JAK3 P52333 4/20 0.41
PTGER1 P34995 2/20 0.40
HTT P42858 2/20 0.38
CA2 P00918 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
TSHR P16473 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17258893 0.87 ALDH1A1 (0.53) TP53GAAKMT2AALDH1A1HPGD
SCHEMBL21048781 0.84 C5AR1 (0.50) GAAKMT2AALDH1A1PTGER1HTT
SCHEMBL21048854 0.84 PTGER1 (0.44) TP53GAAKMT2AALDH1A1HPGD
SCHEMBL17258939 0.79 TP53 (0.50) TP53GAAKMT2AALDH1A1JAK2
SCHEMBL21048978 0.78 TP53 (0.52) TP53GAAKMT2AALDH1A1HPGD
SCHEMBL28840926 0.77 TP53 (0.48) TP53KMT2AJAK2JAK1TYK2
SCHEMBL21048817 0.75 PGR (0.54) GAAKMT2AHPGDPTGER1
SCHEMBL27682450 0.73 ALDH1A1 (0.53) GAAKMT2AALDH1A1HPGDHTT
Hydrochloric Acid SCHEMBL21048875 0.73 ALOX5AP (0.38) KMT2AALDH1A1JAK2JAK1TYK2
SCHEMBL29935885 0.73 CYP1A2 (0.55) GAAKMT2AALDH1A1HPGDHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3143021-B1 PYRAZOLOPYRIDINES AND PYRAZOLOPYRIMIDINES PFIZER (US) 2019-06-12 EP disclosed