SCHEMBL28840926

SCHEMBL28840926

CCCCN(c1ccccc1CNC(=O)O)S(C)(=O)=O

nearest known ligand 0.48

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.48
JAK2 O60674 4/20 0.45
TYK2 P29597 4/20 0.45
JAK3 P52333 4/20 0.45
JAK1 P23458 3/20 0.45
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
PTGER1 P34995 2/20 0.41
ESR1 P03372 1/20 0.40
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17258939 0.92 TP53 (0.50) TP53JAK2TYK2JAK3JAK1
SCHEMBL21048978 0.87 TP53 (0.52) TP53JAK2TYK2JAK3JAK1
SCHEMBL21048878 0.84 JAK2 (0.44) TP53JAK2TYK2JAK3JAK1
SCHEMBL17258776 0.83 JAK2 (0.42) TP53JAK2TYK2JAK3JAK1
SCHEMBL21048854 0.81 PTGER1 (0.44) TP53JAK2TYK2JAK3JAK1
SCHEMBL17258893 0.78 ALDH1A1 (0.53) TP53JAK2MEN1KMT2AL3MBTL1
SCHEMBL21048813 0.77 TP53 (0.41) TP53JAK2TYK2JAK3JAK1
Trifluoroacetic Acid SCHEMBL17258792 0.77 JAK2 (0.40) JAK2TYK2JAK3JAK1MEN1
SCHEMBL17258976 0.76 TP53 (0.42) TP53JAK2TYK2JAK3MEN1
SCHEMBL21048938 0.73 RECQL (0.40) TP53MEN1KMT2AL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106459048-A Pyrazolopyridines and pyrazolopyrimidines 辉瑞公司 2017-02-22 CN disclosed