SCHEMBL21089018

SCHEMBL21089018

CCCCc1ncc(S(C)(=O)=O)cc1N1CC(F)(F)C1

nearest known ligand 0.32

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
CNR2 P34972 4/20 0.31
KDM4E B2RXH2 1/20 0.30
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17196470 0.87 CNR2 (0.33) CNR2
SCHEMBL17177771 0.79 PDE10A (0.33) PTGS2CNR2
SCHEMBL21089051 0.73 ALDH1A1 (0.42) ALOX5PTGS1PTGS2
SCHEMBL21089255 0.69 CTSS (0.36) ALOX5NPC1RAB9A
SCHEMBL17196425 0.62 HRH4 (0.36) PTGS1PTGS2
SCHEMBL21089369 0.61 APLNR (0.34)
SCHEMBL16511461 0.60 ALDH1A1 (0.45) PTGS1PTGS2NPC1
SCHEMBL24587389 0.60 NR1H2 (0.37) CNR2
SCHEMBL17173648 0.60 PTGS2 (0.37) PTGS1PTGS2
SCHEMBL21653458 0.60 TDP1 (0.44) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3495360-A1 HETEROARYL SUBSTITUTED HETEROCYCLYL SULFONES Grünenthal GmbH (DE) 2019-06-12 EP disclosed