SCHEMBL21089283

SCHEMBL21089283

Cc1ccc(CN2CC3(CC(N(C(=O)C(F)(F)F)C4CC4)C3)C2)c(Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.40
CHRM2 P08172 2/20 0.40
CACNA1F O60840 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD2 P14416 1/20 0.40
DRD1 P21728 1/20 0.40
DRD4 P21917 1/20 0.40
ADRA1D P25100 1/20 0.40
HTR7 P34969 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
DRD3 P35462 1/20 0.40
OPRD1 P41143 1/20 0.40
OPRK1 P41145 1/20 0.40
OPRL1 P41146 1/20 0.40
CACNA1D Q01668 1/20 0.40
CACNA1S Q13698 1/20 0.40
CACNA1C Q13936 1/20 0.40
FAAH O00519 4/20 0.37
MGLL Q99685 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21088780 0.90 POLB (0.39) FAAHMGLLP2RX7USP2ALDH1A1
SCHEMBL21088529 0.76 ALDH1A1 (0.43) USP2CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL21089303 0.75 KDM4E (0.43) CYP3A4ALDH1A1
SCHEMBL25924019 0.74
SCHEMBL21088839 0.73 KDM1A (0.41) MGLLUSP2CYP1A2CYP3A4CYP2C9
SCHEMBL21088397 0.73 USP2 (0.36) FAAHMGLLUSP2CYP1A2CYP3A4
SCHEMBL20106999 0.72 CYP3A4 (0.32) CYP3A4
SCHEMBL21088969 0.72 OPRM1 (0.42) OPRM1CHRM2CACNA1FCHRM1DRD2
SCHEMBL20106745 0.71 ITGB3 (0.30)
SCHEMBL21088402 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286172-B1 LSD1 INHIBITORS AND USES THEREOF CONSTELLATION PHARMACEUTICALS INC (US) 2019-06-12 EP disclosed