SCHEMBL21089313

SCHEMBL21089313

CC(C)(C)OC(=O)CCN1CC2(CC(NC3CC3)C2)C1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 2/20 0.35
CNR1 P21554 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.33
CTSK P43235 2/20 0.31
CCR2 P41597 1/20 0.31
DRD2 P14416 1/20 0.31
KCNA3 P22001 1/20 0.31
KDM1A O60341 3/20 0.30
CACNA1H O95180 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21088467 0.87 CNR1 (0.37) EPHX2CNR1SMN1; SMN2CTSKDRD2
SCHEMBL21088332 0.79 EPHX2 (0.33) EPHX2CNR1SMN1; SMN2
SCHEMBL21088777 0.79 KDM1A (0.40) KDM1A
SCHEMBL25923992 0.77 L3MBTL1 (0.40) SMN1; SMN2KDM1A
SCHEMBL20106807 0.76 EHMT2 (0.44) EPHX2SMN1; SMN2CCR2
SCHEMBL21088950 0.73 DRD2 (0.31) DRD2KDM1A
SCHEMBL25924094 0.72 OPRM1 (0.30)
SCHEMBL25923869 0.72 NPSR1 (0.33) KDM1A
SCHEMBL20107004 0.72 KDM1A (0.30) KDM1A
SCHEMBL20106792 0.72 KDM1A (0.44) KDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3286172-B1 LSD1 INHIBITORS AND USES THEREOF CONSTELLATION PHARMACEUTICALS INC (US) 2019-06-12 EP disclosed