SCHEMBL21117864

SCHEMBL21117864

CCOC(=O)[C@H](N)Cc1cccc(C)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
TP53 P04637 1/20 0.50
POLB P06746 1/20 0.47
SLC7A5 Q01650 5/20 0.47
KMT2A Q03164 2/20 0.45
IDO1 P14902 2/20 0.45
MAOB P27338 2/20 0.44
NOS3 P29474 1/20 0.44
NOS1 P29475 1/20 0.44
NOS2 P35228 1/20 0.44
HPGD P15428 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
MEN1 O00255 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
TACR1 P25103 2/20 0.43
KDM4E B2RXH2 1/20 0.43
MAPT P10636 1/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27762534 1.00 ALDH1A1 (0.50) ALDH1A1TP53POLBSLC7A5KMT2A
SCHEMBL20543766 1.00 ALDH1A1 (0.50) ALDH1A1TP53POLBSLC7A5KMT2A
SCHEMBL19699296 0.88 SLC7A5 (0.54) ALDH1A1TP53POLBSLC7A5IDO1
SCHEMBL28637433 0.88 SLC7A5 (0.54) ALDH1A1TP53POLBSLC7A5IDO1
SCHEMBL6218675 0.88 SLC7A5 (0.54) ALDH1A1TP53POLBSLC7A5IDO1
SCHEMBL13588335 0.87 POLB (0.60) ALDH1A1TP53POLBSLC7A5IDO1
SCHEMBL13535116 0.87 POLB (0.60) ALDH1A1TP53POLBSLC7A5IDO1
SCHEMBL2038370 0.86 GRIA2 (0.55) SLC7A5NOS3NOS1NOS2
Hydrochloric Acid SCHEMBL32677180 0.86 SLC7A5 (0.52) ALDH1A1TP53POLBSLC7A5IDO1
Hydrochloric Acid SCHEMBL32676955 0.86 SLC7A5 (0.52) ALDH1A1TP53POLBSLC7A5IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10669242-B2 Clostridium difficile toxin inhibitors Venenum Biodesign, LLC (US) 2020-06-02 US disclosed
US-20190194147-A1 Novel Clostridium Difficile Toxin Inhibitors Venenum Biodesign, LLC (US) 2019-06-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190194147-A1 Novel Clostridium Difficile Toxin Inhibitors GABRA5, GABRA1, GABRA4 ALDH1A1 2381/4885TP53 4810/4885POLB 4138/4885
US-10669242-B2 Clostridium difficile toxin inhibitors GABRA5, GABRA1, GABBR2 ALDH1A1 1908/4885TP53 4770/4885POLB 3866/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.