SCHEMBL21133718

SCHEMBL21133718

C=C/C=C(\C=C/C)C(c1ccccc1)N1CC(CC)(OC)C1

nearest known ligand 0.32

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 6/20 0.32
OPRK1 P41145 6/20 0.32
OPRL1 P41146 6/20 0.32
OPRD1 P41143 7/20 0.31
CYP3A4 P08684 2/20 0.31
CYP2D6 P10635 2/20 0.31
HIF1A Q16665 1/20 0.31
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
KMT2A Q03164 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL70986 0.73 OPRM1 (0.49) OPRM1OPRK1OPRL1OPRD1CYP3A4
SCHEMBL18924468 0.68 ADRA2A (0.35) HIF1AALDH1A1LMNACYP2C19
SCHEMBL20198149 0.68 MGLL (0.48)
SCHEMBL18924436 0.66 HPGD (0.40) HIF1AALDH1A1LMNACYP2C19
SCHEMBL22787085 0.66 ALDH1A1 (0.36) ALDH1A1LMNACYP2C19
SCHEMBL25874874 0.63 HCAR2 (0.40) CYP2D6LMNAKMT2ACYP2C19
SCHEMBL19591149 0.61 OPRK1 (0.38) OPRM1OPRK1OPRL1OPRD1CYP3A4
SCHEMBL19591157 0.61 OPRK1 (0.38) OPRM1OPRK1OPRL1OPRD1CYP3A4
SCHEMBL24310267 0.61 HPGD (0.39) CYP3A4CYP2D6MEN1KMT2A
SCHEMBL17542448 0.61 OPRM1 (0.50) OPRM1OPRK1OPRL1OPRD1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3110816-B1 N2-PHENYL-PYRIDO[3,4-D]PYRIMIDINE-2,8-DIAMINE DERIVATIVES AND THEIR USE AS MPS1 INHIBITORS CANCER RESEARCH TECH LTD (GB) 2019-06-19 EP disclosed