SCHEMBL21153337

SCHEMBL21153337

COc1cc(OC)c(Cl)c(-c2ccc3nc(N)ncc3c2)c1C

nearest known ligand 0.57

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 14/20 0.57
LCK P06239 6/20 0.48
KIT P10721 5/20 0.48
SRC P12931 5/20 0.48
KDR P35968 1/20 0.48
JAK3 P52333 1/20 0.48
MAPK14 Q16539 1/20 0.48
FGFR1 P11362 6/20 0.48
FGFR2 P21802 4/20 0.48
FGFR3 P22607 4/20 0.48
RPS6KB2 Q9UBS0 1/20 0.46
CYP1A2 P05177 1/20 0.44
CSF1R P07333 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19943434 0.94 LCK (0.53) FGFR4LCKKITSRCKDR
SCHEMBL16676911 0.92 FGFR4 (0.66) FGFR4LCKKITSRCKDR
SCHEMBL21153921 0.88 FGFR4 (0.60) FGFR4FGFR1FGFR2FGFR3RPS6KB2
SCHEMBL21154002 0.88 FGFR4 (0.60) FGFR4FGFR1FGFR2FGFR3RPS6KB2
SCHEMBL21153647 0.85 FGFR4 (0.54) FGFR4LCKKITSRCKDR
SCHEMBL22781190 0.84 FGFR4 (0.56) FGFR4LCKKITSRCFGFR1
SCHEMBL21154011 0.83 FGFR4 (0.55) FGFR4FGFR1FGFR2FGFR3RPS6KB2
SCHEMBL21153989 0.83 LCK (0.47) FGFR4LCKKITSRCKDR
SCHEMBL21154059 0.83 FGFR4 (0.56) FGFR4FGFR1FGFR2FGFR3RPS6KB2
SCHEMBL21153914 0.82 FGFR4 (0.51) FGFR4LCKKITSRCKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3508482-B1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR AND USE THEREOF NANJING TRANSTHERA BIOSCIENCES CO LTD (CN) 2020-12-16 EP disclosed
EP-3508482-A1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR AND USE THEREOF Nanjing Transthera Biosciences Co. Ltd. (CN) 2019-07-10 EP disclosed