SCHEMBL21153989

SCHEMBL21153989

CCc1c(OC)cc(OC)c(C)c1-c1ccc2nc(N)ncc2c1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LCK P06239 11/20 0.47
KIT P10721 10/20 0.47
SRC P12931 10/20 0.47
KDR P35968 7/20 0.46
JAK3 P52333 3/20 0.46
MAPK14 Q16539 1/20 0.46
JAK2 O60674 2/20 0.43
JAK1 P23458 2/20 0.43
TYK2 P29597 2/20 0.43
AURKB Q96GD4 2/20 0.43
FGFR4 P22455 1/20 0.41
BRAF P15056 2/20 0.41
DHFR P00374 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19943434 0.89 LCK (0.53) LCKKITSRCKDRJAK3
SCHEMBL21153647 0.87 FGFR4 (0.54) LCKKITSRCKDRJAK3
SCHEMBL19943152 0.86 KDM4E (0.47) FGFR4
SCHEMBL21153337 0.83 FGFR4 (0.57) LCKKITSRCKDRJAK3
SCHEMBL16676911 0.78 FGFR4 (0.66) LCKKITSRCKDRJAK3
SCHEMBL5489026 0.77 LCK (0.55) LCKKITSRCKDRJAK3
SCHEMBL22781316 0.76 FGFR4 (0.52) LCKKITSRCFGFR4
SCHEMBL22781190 0.75 FGFR4 (0.56) LCKKITSRCFGFR4
SCHEMBL21154011 0.74 FGFR4 (0.55) FGFR4
SCHEMBL21154059 0.74 FGFR4 (0.56) FGFR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3508482-A1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR AND USE THEREOF Nanjing Transthera Biosciences Co. Ltd. (CN) 2019-07-10 EP disclosed