SCHEMBL22781190

SCHEMBL22781190

CCCOc1cc(OC)c(Cl)c(-c2ccc3nc(N)ncc3c2)c1Cl

nearest known ligand 0.56

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
FGFR4 P22455 16/20 0.56
FGFR1 P11362 6/20 0.47
FGFR2 P21802 4/20 0.47
FGFR3 P22607 4/20 0.47
RPS6KB2 Q9UBS0 1/20 0.46
LCK P06239 2/20 0.43
KIT P10721 2/20 0.43
SRC P12931 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16676911 0.91 FGFR4 (0.66) FGFR4FGFR1FGFR2FGFR3RPS6KB2
SCHEMBL21153647 0.85 FGFR4 (0.54) FGFR4FGFR1FGFR2FGFR3RPS6KB2
SCHEMBL21153337 0.84 FGFR4 (0.57) FGFR4FGFR1FGFR2FGFR3RPS6KB2
SCHEMBL19943434 0.80 LCK (0.53) FGFR4LCKKITSRC
SCHEMBL21153914 0.79 FGFR4 (0.51) FGFR4FGFR1FGFR2FGFR3RPS6KB2
SCHEMBL29385382 0.78 FGFR4 (0.69) FGFR4FGFR1FGFR2FGFR3RPS6KB2
SCHEMBL15412791 0.78 FGFR4 (0.69) FGFR4FGFR1FGFR2FGFR3RPS6KB2
SCHEMBL16683513 0.77 FGFR4 (0.67) FGFR4FGFR1FGFR2FGFR3RPS6KB2
SCHEMBL5489026 0.76 LCK (0.55) FGFR4LCKKITSRC
SCHEMBL21153989 0.75 LCK (0.47) FGFR4LCKKITSRC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3508482-B1 INHIBITORS OF FIBROBLAST GROWTH FACTOR RECEPTOR AND USE THEREOF NANJING TRANSTHERA BIOSCIENCES CO LTD (CN) 2020-12-16 EP disclosed