SCHEMBL21246424

SCHEMBL21246424

C[C@@H](O)[C@@H](C(=O)NCc1ccc(C(F)(F)F)cc1)N1CC2(CCCCC2)CC1=O

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.40
KCNH2 Q12809 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
NR3C2 P08235 1/20 0.37
CCR2 P41597 5/20 0.36
MTOR P42345 1/20 0.36
CYP2D6 P10635 1/20 0.36
LSS P48449 1/20 0.36
EPHX2 P34913 1/20 0.35
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35
PTGER4 P35408 1/20 0.35
PTGES O14684 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21246426 0.89 GAA (0.41)
SCHEMBL21246427 0.87 SLC1A2 (0.47)
SCHEMBL21246428 0.85 LMNA (0.48)
SCHEMBL21246362 0.82 LMNA (0.46) EPHX2
SCHEMBL21246341 0.81 LMNA (0.48) CYP2D6
SCHEMBL21246364 0.80 CYP3A4 (0.41) NR3C2
SCHEMBL21246359 0.80 SLC1A2 (0.51)
SCHEMBL21246349 0.79 USP19 (0.33)
SCHEMBL21246342 0.78 CYP3A4 (0.43)
SCHEMBL21246360 0.78 USP19 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019152688-A1 SPIRO-LACTAM NMDA RECEPTOR MODULATORS AND USES THEREOF APTINYX INC. (US) 2019-08-08 WO disclosed