SCHEMBL21290177

SCHEMBL21290177

COc1cc(-c2ccccc2)ncc1B1OC(C)(C)C(C)(C)O1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.45
TDO2 P48775 2/20 0.45
DGAT1 O75907 1/20 0.44
SMN1; SMN2 Q16637 5/20 0.43
NPC1 O15118 3/20 0.43
RAB9A P51151 3/20 0.43
ALDH1A1 P00352 3/20 0.43
MAPT P10636 2/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
LPL P06858 1/20 0.42
LIPG Q9Y5X9 1/20 0.42
HPGD P15428 2/20 0.41
LMNA P02545 1/20 0.41
EGFR P00533 1/20 0.40
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
TSHR P16473 2/20 0.40
ATM Q13315 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23956204 0.92 LIPG (0.41) IDO1TDO2DGAT1SMN1; SMN2NPC1
SCHEMBL18015456 0.83 LPL (0.46) IDO1TDO2DGAT1SMN1; SMN2NPC1
SCHEMBL18015448 0.82 LDHA (0.47) IDO1TDO2DGAT1SMN1; SMN2NPC1
SCHEMBL21290169 0.79 NPC1 (0.52) IDO1TDO2DGAT1SMN1; SMN2NPC1
SCHEMBL21290171 0.79 TOP1 (0.46) TDO2DGAT1SMN1; SMN2NPC1RAB9A
SCHEMBL21290170 0.78 ALDH1A1 (0.41) IDO1TDO2DGAT1SMN1; SMN2NPC1
SCHEMBL31642363 0.77 EGFR (0.42) DGAT1LPLLIPGEGFR
SCHEMBL31672743 0.77 EGFR (0.44) DGAT1SMN1; SMN2NPC1RAB9AALDH1A1
SCHEMBL21290090 0.77 DGAT1 (0.46) IDO1TDO2DGAT1SMN1; SMN2NPC1
SCHEMBL20532210 0.76 LPL (0.42) DGAT1SMN1; SMN2NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3752512-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2023-03-01 EP disclosed
EP-3601304-B1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2021-10-27 EP disclosed
WO-2019158453-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2019-08-22 WO disclosed