SCHEMBL2135232

SCHEMBL2135232

CCOC(=O)/C=C/c1cc(OC)ccc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 2/20 0.48
JUN P05412 1/20 0.48
NFKB1 P19838 1/20 0.48
FBP1 P09467 1/20 0.47
CYP3A4 P08684 2/20 0.47
NFE2L2 Q16236 1/20 0.47
FDPS P14324 1/20 0.46
TDP1 Q9NUW8 1/20 0.46
TTR P02766 1/20 0.46
DPP4 P27487 1/20 0.46
ATM Q13315 1/20 0.46
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
CASP3 P42574 1/20 0.45
SENP7 Q9BQF6 1/20 0.45
SENP6 Q9GZR1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16318865 1.00 MAOB (0.48) MAOBJUNNFKB1FBP1CYP3A4
SCHEMBL13686175 0.89 CYP1A2 (0.51) MAOBCYP3A4FDPSTTRDPP4
SCHEMBL1587040 0.89 CYP1A2 (0.51) MAOBCYP3A4FDPSTTRDPP4
SCHEMBL2325706 0.85 CYP3A4 (0.51) MAOBCYP3A4NFE2L2FDPSTTR
SCHEMBL31390627 0.85 CYP3A4 (0.51) MAOBCYP3A4NFE2L2FDPSTTR
SCHEMBL2325697 0.85 CYP3A4 (0.51) MAOBCYP3A4NFE2L2FDPSTTR
SCHEMBL19257215 0.83 MAOB (0.48) MAOBJUNNFKB1FBP1CYP3A4
SCHEMBL31462784 0.83 MAPT (0.49) MAOBCYP3A4FDPSTTRDPP4
SCHEMBL29090924 0.83 MAOB (0.51) MAOBJUNNFKB1NFE2L2ATM
SCHEMBL4592405 0.82 MAPT (0.68) MAOBCYP3A4TDP1CYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9181186-B2 Aromatic ring compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-11-10 US disclosed
US-20150045378-A1 AROMATIC RING COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2015-02-12 US disclosed
EP-2816032-A1 AROMATIC RING COMPOUND Takeda Pharmaceutical Company Limited (JP) 2014-12-24 EP disclosed
US-20120101105-A1 ARYL SUBSTITUTED CARBOXAMIDE DERIVATIVES AS CALCIUM OR SODIUM CHANNEL BLOCKERS RAQUALIA PHARMA INC. (JP) 2012-04-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120101105-A1 ARYL SUBSTITUTED CARBOXAMIDE DERIVATIVES AS CALCIUM OR SODIUM CHANNEL BLOCKERS CACNA1I, CACNA1G, CACNA1H MAOB 1156/4885JUN 3173/4885NFKB1 1234/4885
US-20150045378-A1 AROMATIC RING COMPOUND GPR119, GPR27, GPR4 MAOB 3876/4885JUN 1588/4885NFKB1 953/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.