SCHEMBL21362417

SCHEMBL21362417

CCC(C)Cc1ccc(C(=O)c2ccc(F)cc2)c(Br)c1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNA7 P36544 2/20 0.38
ALDH1A1 P00352 4/20 0.38
LMNA P02545 3/20 0.38
GAA P10253 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
EPHX2 P34913 1/20 0.36
PPARG P37231 1/20 0.36
THRB P10828 1/20 0.35
HPGD P15428 1/20 0.35
MAPT P10636 2/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
TRPA1 O75762 1/20 0.34
S1PR1 P21453 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157516 0.84 ALDH1A1 (0.48) CHRNA7ALDH1A1LMNAGAATDP1
SCHEMBL21362526 0.81 CHRNA7 (0.35) CHRNA7ALDH1A1LMNAHPGDMAPT
SCHEMBL21362558 0.81 DPP4 (0.40) ALDH1A1LMNAGAATDP1THRB
SCHEMBL20157552 0.80 LMNA (0.38) CHRNA7ALDH1A1LMNAGAATHRB
SCHEMBL20157553 0.80 POLB (0.36) CHRNA7ALDH1A1LMNAGAATHRB
SCHEMBL20157560 0.79 PTPN1 (0.43) ALDH1A1LMNAGAAMAPTHTT
SCHEMBL21362538 0.79 SRD5A2 (0.39) CHRNA7ALDH1A1LMNAGAATDP1
SCHEMBL1252299 0.78 GAA (0.50) CHRNA7ALDH1A1LMNAGAATHRB
SCHEMBL20157579 0.78 TP53 (0.38) CHRNA7ALDH1A1LMNAGAATDP1
SCHEMBL21362418 0.78 THRA (0.47) PPARGTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed