SCHEMBL21362418

SCHEMBL21362418

CCCCCc1ccc(C(=O)c2ccc(F)cc2)c(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
THRA P10827 3/20 0.47
THRB P10828 3/20 0.47
PPARA Q07869 2/20 0.47
RARB P10826 7/20 0.46
RARA P10276 1/20 0.46
RARG P13631 1/20 0.46
PPARG P37231 1/20 0.44
KAT8 Q9H7Z6 2/20 0.44
HTR7 P34969 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157516 0.85 ALDH1A1 (0.48) THRB
SCHEMBL6936245 0.82 THRA (0.56) THRATHRBRARBRARA
SCHEMBL21362558 0.82 DPP4 (0.40) THRATHRB
SCHEMBL20157560 0.80 PTPN1 (0.43)
SCHEMBL21362538 0.80 SRD5A2 (0.39) THRB
SCHEMBL1252299 0.79 GAA (0.50) THRB
SCHEMBL20157579 0.79 TP53 (0.38) THRB
SCHEMBL20157580 0.79 LMNA (0.37) THRB
SCHEMBL11871709 0.79 PPARA (0.68) PPARARARBRARARARGPPARG
SCHEMBL20157757 0.78 LMNA (0.50) THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed