SCHEMBL21362558

SCHEMBL21362558

CC(C)CCc1ccc(C(=O)c2ccc(F)cc2)c(Br)c1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.40
GRIN2D O15399 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
S1PR1 P21453 1/20 0.37
HPGD P15428 2/20 0.37
ALDH1A1 P00352 5/20 0.36
LMNA P02545 4/20 0.36
GAA P10253 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
MAPK14 Q16539 1/20 0.36
MAPT P10636 2/20 0.35
PRNP P04156 1/20 0.35
THRB P10828 2/20 0.35
THRA P10827 1/20 0.35
CES2 O00748 1/20 0.35
CES1 P23141 1/20 0.35
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20157516 0.82 ALDH1A1 (0.48) ALDH1A1LMNAGAATDP1MAPT
SCHEMBL21362418 0.82 THRA (0.47) THRBTHRA
SCHEMBL20157552 0.81 LMNA (0.38) S1PR1ALDH1A1LMNAGAAMAPT
SCHEMBL21362417 0.81 CHRNA7 (0.38) S1PR1HPGDALDH1A1LMNAGAA
SCHEMBL20157553 0.81 POLB (0.36) S1PR1HPGDALDH1A1LMNAGAA
SCHEMBL20157560 0.80 PTPN1 (0.43) S1PR1ALDH1A1LMNAGAAMAPT
SCHEMBL20157757 0.78 LMNA (0.50) S1PR1ALDH1A1LMNAGAAMAPT
SCHEMBL20157523 0.78 CES2 (0.39) S1PR1ALDH1A1LMNAGAAMAPT
SCHEMBL21362538 0.77 SRD5A2 (0.39) S1PR1ALDH1A1LMNAGAATDP1
SCHEMBL20157557 0.77 PTPN1 (0.39) S1PR1ALDH1A1LMNAGAAMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3539960-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF Luoxin Pharmaceutical (Shanghai) Co., Ltd. (CN) 2019-09-18 EP disclosed