SCHEMBL20158023

SCHEMBL20158023

COc1cc(C)ccc1C(=O)c1ccc(CBr)cc1Br

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.45
RIN1 Q13671 1/20 0.45
L3MBTL1 Q9Y468 5/20 0.40
SMN1; SMN2 Q16637 4/20 0.40
MAPT P10636 4/20 0.40
ALDH1A1 P00352 3/20 0.40
HPGD P15428 3/20 0.40
IDO1 P14902 1/20 0.39
TDO2 P48775 1/20 0.39
LCK P06239 1/20 0.39
FYN P06241 1/20 0.39
NPC1 O15118 2/20 0.38
CYP4F2 P78329 1/20 0.38
CYP4A11 Q02928 1/20 0.38
ACHE P22303 1/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20158021 0.87 LCK (0.46) ABL1RIN1L3MBTL1SMN1; SMN2MAPT
SCHEMBL20157512 0.85 NPC1 (0.46) SMN1; SMN2MAPTALDH1A1LCKFYN
SCHEMBL20157821 0.81 CYP4F2 (0.46) SMN1; SMN2MAPTALDH1A1HPGDNPC1
SCHEMBL20157772 0.81 LOXL2 (0.38) ABL1RIN1MAPTALDH1A1NPC1
SCHEMBL21362819 0.80 ACHE (0.40) SMN1; SMN2ALDH1A1LCKFYNNPC1
SCHEMBL20157609 0.79 ALDH1A1 (0.46) MAPTALDH1A1HPGDNPC1ACHE
SCHEMBL20157960 0.79 SRD5A2 (0.49) L3MBTL1MAPTALDH1A1NPC1CYP4F2
SCHEMBL20158157 0.78 KMT2A (0.41) ABL1RIN1L3MBTL1SMN1; SMN2MAPT
SCHEMBL7577375 0.77 CYP4F2 (0.44) ABL1RIN1L3MBTL1SMN1; SMN2MAPT
SCHEMBL20157984 0.77 NPC1 (0.38) SMN1; SMN2MAPTALDH1A1HPGDLCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018086605-A1 NITROGENOUS MACROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR, PHARMACEUTICAL COMPOSITION AND APPLICATION THEREOF 山东罗欣药业集团股份有限公司 2018-05-17 WO disclosed