SCHEMBL21363516

SCHEMBL21363516

OC(c1ccc(Cl)cc1)C1CCO1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.38
HSD17B2 P37059 1/20 0.35
HPGD P15428 2/20 0.35
GAA P10253 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
BCL2A1 Q16548 1/20 0.35
TSHR P16473 2/20 0.34
MAPK1 P28482 2/20 0.34
HIF1A Q16665 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
SLC6A3 Q01959 5/20 0.34
FPR2 P25090 2/20 0.33
PROKR1 Q8TCW9 2/20 0.33
AOC3 Q16853 1/20 0.33
SLC6A2 P23975 1/20 0.33
SLC6A4 P31645 1/20 0.33
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
ADRB2 P07550 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1128830 0.90 SLC6A3 (0.45) RAB9AHPGDGAASMN1; SMN2TDP1
SCHEMBL16861575 0.76 BCL2A1 (0.49) HPGDBCL2A1TSHRFPR2PROKR1
SCHEMBL1349046 0.75 FPR2 (0.45) HSD17B2HPGDGAASMN1; SMN2TSHR
SCHEMBL1237578 0.73 POLB (0.42) RAB9ASLC6A3LMNAALDH1A1
Cyclopropane SCHEMBL6425247 0.72 DHODH (0.47) HSD17B2HPGDGAASMN1; SMN2SLC6A3
SCHEMBL8611840 0.72 DHODH (0.51) RAB9AHPGDGAASMN1; SMN2SLC6A3
SCHEMBL10749366 0.72 DHODH (0.47) HSD17B2HPGDGAASMN1; SMN2SLC6A3
SCHEMBL11348436 0.72 SLC6A3 (0.50) HPGDGAASMN1; SMN2TDP1SLC6A3
SCHEMBL9891700 0.72 SLC6A3 (0.40) HPGDSMN1; SMN2SLC6A3ALDH1A1
SCHEMBL5415203 0.71 DRD4 (0.56) TSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11655245-B2 Oxadiazole transient receptor potential channel inhibitors GENENTECH, INC. (US) 2023-05-23 US disclosed
US-20230121700-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS GENENTECH, INC. (US) 2023-04-20 US disclosed
US-20200308161-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS GENENTECH, INC. (US) 2020-10-01 US disclosed
US-10710994-B2 Oxadiazole transient receptor potential channel inhibitors GENENTECH, INC. (US) 2020-07-14 US disclosed
US-20190284179-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS GENENTECH, INC. (US) 2019-09-19 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11655245-B2 Oxadiazole transient receptor potential channel inhibitors TRPA1, TRPV1, P2RX3 RAB9A 3715/4885HSD17B2 3016/4885HPGD 822/4885
US-20190284179-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS TRPA1, TRPV1, TRPV3 RAB9A 3728/4885HSD17B2 2760/4885HPGD 816/4885
US-20200308161-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS TRPA1, TRPV1, P2RX3 RAB9A 3715/4885HSD17B2 3016/4885HPGD 822/4885
US-10710994-B2 Oxadiazole transient receptor potential channel inhibitors TRPA1, TRPV1, TRPV3 RAB9A 3728/4885HSD17B2 2760/4885HPGD 816/4885
US-20230121700-A1 OXADIAZOLE TRANSIENT RECEPTOR POTENTIAL CHANNEL INHIBITORS TRPA1, TRPV1, TRPV3 RAB9A 3728/4885HSD17B2 2760/4885HPGD 816/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.