SCHEMBL21384573

SCHEMBL21384573

CCOC(=O)C(C)C1CCN(c2ccc(OC)cc2)CC1

nearest known ligand 0.54

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
GAA P10253 2/20 0.54
L3MBTL1 Q9Y468 1/20 0.48
POLB P06746 2/20 0.47
MAPK1 P28482 1/20 0.47
MAPT P10636 5/20 0.47
KMT2A Q03164 5/20 0.47
MEN1 O00255 3/20 0.47
GFER P55789 2/20 0.46
DRD2 P14416 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.45
THRB P10828 1/20 0.45
NR4A1 P22736 1/20 0.45
RAB9A P51151 1/20 0.45
MCL1 Q07820 1/20 0.45
AKR1C3 P42330 1/20 0.45
ACACB O00763 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28452277 0.86 ALDH1A1 (0.53) ALDH1A1GAAL3MBTL1POLBMAPK1
SCHEMBL21385141 0.85 MAPT (0.45) ALDH1A1GAAL3MBTL1POLBMAPT
SCHEMBL21384617 0.85 L3MBTL1 (0.51) ALDH1A1GAAL3MBTL1POLBMAPK1
SCHEMBL10685927 0.83 GAA (0.50) ALDH1A1GAAL3MBTL1POLBMAPK1
SCHEMBL21384587 0.82 CHRNB2 (0.47) ACACB
SCHEMBL3139067 0.81 MAPT (0.67) ALDH1A1GAAL3MBTL1POLBMAPK1
SCHEMBL3225431 0.81 CCR1 (0.52) MAPK1MAPT
SCHEMBL17730831 0.80 ALDH1A1 (0.46) ALDH1A1GAAMAPTKMT2AMEN1
SCHEMBL12988256 0.78 HTR3E (0.54) ALDH1A1GAAL3MBTL1POLBMAPK1
SCHEMBL21384585 0.77 L3MBTL1 (0.49) ALDH1A1GAAL3MBTL1POLBMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117185987-A Amidine and guanidine derivatives, preparation method and medical application thereof 四川科伦博泰生物医药股份有限公司 2023-12-08 CN disclosed
CN-111630048-B Amidine and guanidine derivatives, preparation method and medical application thereof 四川科伦博泰生物医药股份有限公司 2023-09-29 CN disclosed
CN-111630048-A Amidine and guanidine derivatives, preparation method and application thereof in medicines 四川科伦博泰生物医药股份有限公司 2020-09-04 CN disclosed
WO-2019179362-A1 AMIDINE AND GUANIDINE DERIVATIVES, PREPARATION METHOD THEREFOR AND MEDICAL USES THEREOF 四川科伦博泰生物医药股份有限公司 2019-09-26 WO disclosed