SCHEMBL21391072

SCHEMBL21391072

COc1ccc2nc(CCCC(=O)CC(C)(O)c3ccccc3)n(C3CCC3)c2n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 9/20 0.34
CYP11B2 P19099 1/20 0.34
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
ACSS2 Q9NR19 1/20 0.31
MTNR1A P48039 1/20 0.31
MTNR1B P49286 1/20 0.31
OPRM1 P35372 1/20 0.31
OPRD1 P41143 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21391130 0.89 CYP11B2 (0.38) PDE10ACYP11B2PIK3CAMTOR
SCHEMBL21391133 0.88 CYP11B1 (0.33) CYP11B2ALDH1A1ACSS2TNKSPARP2
SCHEMBL21391073 0.87 PDE10A (0.37) PDE10ACYP11B2PIK3CAMTOR
SCHEMBL21390955 0.85 ALDH1A1 (0.32) ALDH1A1ACSS2
SCHEMBL21391134 0.84 RORC (0.33) ALDH1A1ACSS2TNKSPARP1PARP2
SCHEMBL21390764 0.83 CYP11B1 (0.35) CYP11B2ALDH1A1ACSS2
SCHEMBL21391070 0.82 CYP11B2 (0.36) PDE10ACYP11B2PIK3CAMTOR
SCHEMBL21390952 0.82 RORC (0.34) ALDH1A1ACSS2TNKSPARP1PARP2
SCHEMBL21391131 0.81 CYP11B2 (0.37) PDE10ACYP11B2ALDH1A1PIK3CAMTOR
SCHEMBL20624369 0.80 ADRB2 (0.37) PDE10ACYP11B2CNR1CNR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183148-A1 KV7 CHANNEL ACTIVATORS COMPOSITIONS AND METHODS OF USE KNOPP BIOSCIENCES LLC (US) 2019-09-26 WO disclosed