SCHEMBL21394569

SCHEMBL21394569

Nc1cc(Cc2cccc(Cl)c2)ccn1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.50
NOS1 P29475 1/20 0.50
NOS2 P35228 1/20 0.50
MPO P05164 2/20 0.49
BACE1 P56817 1/20 0.49
PNMT P11086 2/20 0.48
TAAR1 Q96RJ0 3/20 0.46
GABRP O00591 1/20 0.45
GABRD O14764 1/20 0.45
GABRA1 P14867 1/20 0.45
GABRB1 P18505 1/20 0.45
GABRG2 P18507 1/20 0.45
GABRB3 P28472 1/20 0.45
GABRA5 P31644 1/20 0.45
GABRA3 P34903 1/20 0.45
GABRA2 P47869 1/20 0.45
GABRB2 P47870 1/20 0.45
GABRA4 P48169 1/20 0.45
GABRE P78334 1/20 0.45
GABRA6 Q16445 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL21384143 0.98 NOS1 (0.49) NOS3NOS1NOS2MPOBACE1
SCHEMBL18586524 0.82 MPO (0.55) NOS3NOS1MPOPNMTTAAR1
SCHEMBL1600990 0.82 NOS3 (0.57) NOS3NOS1NOS2MPOTAAR1
SCHEMBL3300276 0.79 PNMT (0.65) PNMTTAAR1CYP3A4IDO1AGXT
SCHEMBL1501368 0.78 ALDH1A1 (0.55) PNMTTAAR1CYP3A4IDO1AGXT
SCHEMBL21384277 0.78 PNMT (0.47) NOS3NOS1MPOBACE1PNMT
SCHEMBL29442853 0.78 PNMT (0.47) NOS3NOS1MPOBACE1PNMT
SCHEMBL21384198 0.77 TP53 (0.55) MPOBACE1PNMTTAAR1CYP3A4
SCHEMBL29442835 0.77 TP53 (0.55) MPOBACE1PNMTTAAR1CYP3A4
SCHEMBL21394729 0.76 TAAR1 (0.42) MPOBACE1PNMTTAAR1HTR3E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed