SCHEMBL21395084

SCHEMBL21395084

Cn1ccc(C(=O)Nc2ccc(Cc3cc(F)cc(F)c3)cn2)nc1=O

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AHR P35869 1/20 0.39
GRM5 P41594 5/20 0.39
NPC1 O15118 1/20 0.39
TSHR P16473 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CYP1A2 P05177 3/20 0.38
CYP2C9 P11712 3/20 0.38
KCNH2 Q12809 1/20 0.38
CYP3A4 P08684 3/20 0.38
SLC6A3 Q01959 1/20 0.38
ABCB1 P08183 2/20 0.36
JAK2 O60674 1/20 0.36
NTRK1 P04629 1/20 0.36
ABCC1 P33527 1/20 0.36
CACNA1H O95180 1/20 0.36
KDM4E B2RXH2 1/20 0.36
GCK P35557 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21395020 0.89 CACNA1H (0.43) AHRGRM5NPC1TSHRRAB9A
SCHEMBL21394958 0.84 P2RX3 (0.42) AHRNPC1TSHRRAB9ASMN1; SMN2
SCHEMBL21394747 0.82 AHR (0.38) AHRGRM5NPC1TSHRRAB9A
SCHEMBL29442838 0.80 RAB9A (0.64) GRM5NPC1TSHRRAB9ASMN1; SMN2
SCHEMBL21394572 0.80 TSHR (0.44) GRM5NPC1TSHRRAB9ASMN1; SMN2
SCHEMBL21394807 0.80 RAB9A (0.64) GRM5NPC1TSHRRAB9ASMN1; SMN2
SCHEMBL29357109 0.80 TSHR (0.44) GRM5NPC1TSHRRAB9ASMN1; SMN2
SCHEMBL21394918 0.80 GRM5 (0.43) GRM5NPC1RAB9ASMN1; SMN2CYP1A2
SCHEMBL21394930 0.79 GRM5 (0.40) GRM5NPC1TSHRRAB9ASMN1; SMN2
SCHEMBL21395129 0.78 GRM5 (0.40) AHRGRM5NPC1TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020198026-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2020-10-01 WO disclosed
WO-2019183587-A1 COMPOUNDS AND USES THEREOF YUMANITY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed