SCHEMBL21397401

SCHEMBL21397401

CCCC1(CCC=N)Cc2ccccc2[C@H]1N

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 2/20 0.31
MAOA P21397 2/20 0.31
MAOB P27338 2/20 0.31
HTR2A P28223 1/20 0.30
ADRA2A P08913 1/20 0.30
ADRA2B P18089 1/20 0.30
ADRA2C P18825 1/20 0.30
ADRA1B P35368 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21397676 1.00 KDM1A (0.31) KDM1AMAOAMAOBHTR2AADRA2A
SCHEMBL21397337 0.89 HTR2A (0.37) KDM1AMAOAMAOBHTR2AADRA2A
SCHEMBL21397653 0.83 HTR2A (0.35) KDM1AMAOAMAOBHTR2AADRA2A
SCHEMBL21397670 0.80 HTR2A (0.33) KDM1AMAOAMAOBHTR2AADRA2A
SCHEMBL21397647 0.78 DRD2 (0.36) KDM1AMAOAMAOBHTR2AADRA2A
SCHEMBL21397678 0.76 HTR2A (0.39) KDM1AHTR2AADRA2AADRA2BADRA2C
SCHEMBL12086608 0.68 SLC10A2 (0.37) KDM1AMAOAMAOBHTR2AADRA2A
SCHEMBL21397675 0.68 HTR2A (0.40) HTR2AADRA2AADRA2BADRA2CADRA1B
SCHEMBL22515436 0.67 ALOX12 (0.38) ADRA2AADRA2BADRA2CADRA1B
SCHEMBL21397500 0.67 ADRA2A (0.35) KDM1AMAOAMAOBHTR2AADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019183367-A1 SHP2 PHOSPHATASE INHIBITORS AND METHODS OF USE THEREOF RELAY THERAPEUTICS, INC. (US) 2019-09-26 WO disclosed