SCHEMBL2145351

SCHEMBL2145351

N#Cc1ccc(OCCn2cnc(C(=O)O)c2O)cc1

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NSD2 O96028 1/20 0.49
NSD3 Q9BZ95 1/20 0.49
TBXAS1 P24557 1/20 0.47
MMP2 P08253 2/20 0.47
KCNA5 P22460 5/20 0.46
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
MMP3 P08254 2/20 0.42
MMP1 P03956 1/20 0.41
MMP9 P14780 1/20 0.41
MMP13 P45452 1/20 0.41
CYP19A1 P11511 3/20 0.41
EIF4EBP1 Q13541 1/20 0.41
LTA4H P09960 2/20 0.41
NTRK1 P04629 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2145277 0.89 NSD2 (0.51) NSD2NSD3TBXAS1MMP2KCNA5
SCHEMBL2145861 0.85 L3MBTL1 (0.52) TBXAS1ALDH1A1LTA4H
SCHEMBL2146065 0.84 GABRA1 (0.48) NSD2NSD3TBXAS1MMP2KCNA5
SCHEMBL2145878 0.84 RXFP1 (0.48) NSD2NSD3TBXAS1ALDH1A1
SCHEMBL2145870 0.80 MAPK1 (0.57) TBXAS1ALDH1A1MAPT
SCHEMBL2145709 0.77 TBXAS1 (0.51) TBXAS1ALDH1A1
SCHEMBL2145381 0.76 NSD2 (0.51) NSD2NSD3TBXAS1MMP2KCNA5
SCHEMBL2145655 0.76 HRH2 (0.45) NSD2NSD3TBXAS1MMP2KCNA5
SCHEMBL2145473 0.75 GAA (0.51) TBXAS1ALDH1A1LTA4H
SCHEMBL2145204 0.74 GABRA1 (0.43) NSD2NSD3TBXAS1MMP2KCNA5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2040702-B1 USE OF AMPK-ACTIVATING IMIDAZOLE DERIVATIVES, PREPARATION PROCESS THEREFOR AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM MERCK PATENT GMBH (DE) 2011-07-27 EP claimed