SCHEMBL2145878

SCHEMBL2145878

O=C(O)c1ncn(CCOc2ccc(F)cc2)c1O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.48
NSD2 O96028 1/20 0.47
NSD3 Q9BZ95 1/20 0.47
IDO1 P14902 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
TBXAS1 P24557 2/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
HTT P42858 2/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 1/20 0.41
GAA P10253 1/20 0.41
CYP2C9 P11712 1/20 0.41
HPGD P15428 1/20 0.41
CYP2C19 P33261 1/20 0.41
KDM4E B2RXH2 1/20 0.41
NR4A2 P43354 1/20 0.40
LMNA P02545 1/20 0.40
MAPK13 O15264 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2145752 0.88 NSD2 (0.49) RXFP1NSD2NSD3IDO1NPC1
SCHEMBL2145861 0.87 L3MBTL1 (0.52) NPC1RAB9ATBXAS1SMN1; SMN2HTT
SCHEMBL2145351 0.84 NSD2 (0.49) NSD2NSD3TBXAS1ALDH1A1
SCHEMBL2145448 0.84 NPC1 (0.49) RXFP1NSD2NSD3NPC1RAB9A
SCHEMBL2145870 0.82 MAPK1 (0.57) NPC1RAB9ATBXAS1SMN1; SMN2HTT
SCHEMBL2145709 0.79 TBXAS1 (0.51) TBXAS1SMN1; SMN2HTTMEN1KMT2A
SCHEMBL2145473 0.77 GAA (0.51) NPC1RAB9ATBXAS1SMN1; SMN2HTT
SCHEMBL2145545 0.75 NSD2 (0.49) RXFP1NSD2NSD3IDO1NPC1
SCHEMBL2145421 0.73 ALDH1A1 (0.42) RXFP1NSD2NSD3NPC1RAB9A
SCHEMBL2145876 0.73 NPC1 (0.47) NPC1RAB9ASMN1; SMN2HTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2040702-B1 USE OF AMPK-ACTIVATING IMIDAZOLE DERIVATIVES, PREPARATION PROCESS THEREFOR AND PHARMACEUTICAL COMPOSITIONS COMPRISING THEM MERCK PATENT GMBH (DE) 2011-07-27 EP claimed