SCHEMBL2145779

SCHEMBL2145779

CCOC(=O)c1sc(C)nc1C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.54
HPGD P15428 3/20 0.54
MAPT P10636 6/20 0.50
POLB P06746 1/20 0.50
NPC1 O15118 1/20 0.49
KDM4E B2RXH2 3/20 0.48
MEN1 O00255 2/20 0.48
KMT2A Q03164 2/20 0.48
HSP90AA1 P07900 1/20 0.48
CRHBP P24387 1/20 0.48
CRHR2 Q13324 1/20 0.48
CYP1A2 P05177 1/20 0.46
GAA P10253 2/20 0.46
TSHR P16473 1/20 0.46
HTT P42858 1/20 0.46
HSD17B10 Q99714 1/20 0.46
P2RY1 P47900 1/20 0.43
LMNA P02545 1/20 0.43
HDAC3 O15379 1/20 0.42
HDAC4 P56524 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL299362 0.86 ALDH1A1 (0.52) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL10821105 0.86 ALDH1A1 (0.52) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL6137641 0.86 ALDH1A1 (0.52) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL9750672 0.86 ALDH1A1 (0.52) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL10242354 0.85 ALDH1A1 (0.72) ALDH1A1HPGDMAPTNPC1KDM4E
SCHEMBL244255 0.84 ALDH1A1 (0.76) ALDH1A1HPGDMAPTNPC1KDM4E
SCHEMBL2309900 0.84 ALDH1A1 (0.51) ALDH1A1HPGDMAPTNPC1KDM4E
SCHEMBL8507216 0.84 ALDH1A1 (0.51) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL3454323 0.84 ALDH1A1 (0.51) ALDH1A1HPGDMAPTKDM4EMEN1
SCHEMBL9287012 0.84 POLB (0.48) ALDH1A1HPGDMAPTPOLBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 62 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119751376-A Preparation method of thifluzamide 广东禾康精细化工有限公司 2025-04-04 CN disclosed
CN-116354902-A Green and environment-friendly process for synthesizing 2-methyl-4-trifluoromethyl-5-thiazole formic acid 广东禾康精细化工有限公司 2023-06-30 CN disclosed
EP-3186227-B1 NOVEL SULFONYLAMINOBENZAMIDE COMPOUNDS AS ANTHELMINTICS ELANCO TIERGESUNDHEIT AG (CH) 2021-03-24 EP disclosed
EP-3792251-A1 NOVEL SULFONYLAMINOBENZAMIDE COMPOUNDS AS ANTHELMINTICS Elanco Tiergesundheit AG (CH) 2021-03-17 EP disclosed
US-10464889-B2 Sulfonylaminobenzamide compounds as anthelmintics ELANCO TIERGESUNDHEIT AG (US) 2019-11-05 US disclosed
US-20180161331-A1 NOVEL TETRAHYDROPYRIDOPYRIMIDINE COMPOUND OR SALT THEREOF TAIHO PHARMACEUTICAL CO., LTD. (JP) 2018-06-14 US disclosed
US-9889136-B2 Tetrahydropyridopyrimidine compound or salt thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2018-02-13 US disclosed
US-20170226053-A1 NOVEL SULFONYLAMINOBENZAMIDE COMPOUNDS AS ANTHELMINTICS NOVARTIS TIERGESUNDHEIT AG (CH) 2017-08-10 US disclosed
US-20170226053-A1 NOVEL SULFONYLAMINOBENZAMIDE COMPOUNDS AS ANTHELMINTICS NOVARTIS TIERGESUNDHEIT AG (CH) 2017-08-10 US disclosed
US-9662333-B2 Tetrahydropyridopyrimidine compound or salt thereof TAIHO PHARMACEUTICAL CO., LTD. (JP) 2017-05-30 US disclosed
EP-0648742-A1 Improved process for the preparation of thioacetamide ROHM AND HAAS COMPANY (US) 1995-04-19 EP disclosed
EP-0371950-B1 Substituted thiazoles and their use as fungicides MONSANTO CO (US) 1995-01-11 EP disclosed
US-5284974-A Reaction of acetonitrile with hydrogen sulfide using a polymer supported amine catalyst MONSANTO COMPANY (US) 1994-02-08 US disclosed
CN-1021010-C SUBSTITUTED THIAZOLES COMPOSITION AND THEIR USE AS FUNGICIDES MONSANTO CO (US) 1993-06-02 CN disclosed
EP-0276177-B1 HETEROCYCLIC DERIVATIVES, METHOD FOR THEIR PREPARATION AND FUNGICIDES CONTAINING THEM AS ACTIVE INGREDIENTS SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1992-01-29 EP disclosed
US-5045554-A Fluoro compounds, rice sheath blight, Basidiomycetes type fungus MONSANTO COMPANY (US) 1991-09-03 US disclosed
CN-1043127-A Substituted thiazole and mycocide purposes thereof MONSANTO CO (US) 1990-06-20 CN disclosed
EP-0371950-A2 Substituted thiazoles and their use as fungicides Monsanto Company (US) 1990-06-06 EP disclosed
US-4837242-A Thiazoles and pyrazoles as fungicides SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1989-06-06 US disclosed
EP-0276177-A1 Heterocyclic derivatives, method for their preparation and fungicides containing them as active ingredients SUMITOMO CHEMICAL COMPANY, LIMITED (JP) 1988-07-27 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20180161331-A1 NOVEL TETRAHYDROPYRIDOPYRIMIDINE COMPOUND OR SALT THEREOF NR5A1, CYP17A1, AR ALDH1A1 295/4885HPGD 208/4885MAPT 2428/4885
US-20170226053-A1 NOVEL SULFONYLAMINOBENZAMIDE COMPOUNDS AS ANTHELMINTICS PKD2, CATSPER1, PKD1 ALDH1A1 1365/4885HPGD 3420/4885MAPT 4755/4885
US-10464889-B2 Sulfonylaminobenzamide compounds as anthelmintics PKD2, CATSPER1, ATP1B2 ALDH1A1 1120/4885HPGD 2857/4885MAPT 4705/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.