SCHEMBL21551957

SCHEMBL21551957

CN1CCN(CCCNC(=O)c2ccc(/C=C/c3cc(Br)cc(Br)c3)cc2)CC1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HDAC2 Q92769 1/20 0.59
HDAC8 Q9BY41 1/20 0.59
HDAC6 Q9UBN7 1/20 0.59
MAPT P10636 3/20 0.55
SMN1; SMN2 Q16637 3/20 0.55
LMNA P02545 2/20 0.55
ALDH1A1 P00352 2/20 0.55
GAA P10253 1/20 0.55
MAPK1 P28482 1/20 0.55
HTT P42858 1/20 0.55
TSHR P16473 1/20 0.55
RAD52 P43351 1/20 0.53
KMT2A Q03164 3/20 0.52
MEN1 O00255 1/20 0.52
DRD2 P14416 3/20 0.50
DRD3 P35462 3/20 0.50
DRD4 P21917 1/20 0.47
TP53 P04637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21551990 0.82 LMNA (0.54) HDAC2HDAC8HDAC6MAPTSMN1; SMN2
SCHEMBL21551981 0.80 LMNA (0.52) HDAC2HDAC8HDAC6MAPTSMN1; SMN2
SCHEMBL21551941 0.80 HDAC6 (0.62) HDAC2HDAC8HDAC6MAPTTSHR
SCHEMBL178534 0.78 KMT2A (0.71) HDAC2HDAC8HDAC6MAPTSMN1; SMN2
SCHEMBL12760681 0.78 MAPT (0.64) HDAC2HDAC8HDAC6MAPTSMN1; SMN2
SCHEMBL16227646 0.77 ALDH1A1 (0.69) HDAC2HDAC8HDAC6MAPTSMN1; SMN2
SCHEMBL21551964 0.77 TSHR (0.54) MAPTSMN1; SMN2LMNAALDH1A1GAA
SCHEMBL19226707 0.76 SMN1; SMN2 (0.92) HDAC2HDAC8HDAC6MAPTSMN1; SMN2
SCHEMBL21551954 0.75 TSHR (0.69) MAPTSMN1; SMN2LMNAALDH1A1MAPK1
SCHEMBL12074931 0.75 LMNA (0.92) HDAC2HDAC8HDAC6MAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019216810-A1 NEW ANTIFUNGAL COMPOUNDS URBAN CONSTANTIN (SE) 2019-11-14 WO claimed
WO-2019216810-A1 NEW ANTIFUNGAL COMPOUNDS URBAN CONSTANTIN (SE) 2019-11-14 WO disclosed