SCHEMBL21590167

SCHEMBL21590167

COc1ccc(S(N)(=O)=O)c(-c2ccc(Br)cc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC8 Q9BY41 1/20 0.47
PTGS2 P35354 2/20 0.44
CA2 P00918 8/20 0.43
CA9 Q16790 7/20 0.43
CA1 P00915 7/20 0.43
CA12 O43570 4/20 0.43
ESR1 P03372 1/20 0.42
ESR2 Q92731 1/20 0.42
ACHE P22303 3/20 0.41
CA14 Q9ULX7 2/20 0.41
PAX8 Q06710 1/20 0.41
CA7 P43166 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
HPGD P15428 1/20 0.40
HTT P42858 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28134928 0.91 PTGS2 (0.44) PTGS2CA2CA9CA1ACHE
Hydrochloric Acid SCHEMBL5797690 0.84 PTGS2 (0.45) PTGS2CA2CA9CA1CA12
SCHEMBL16936936 0.80 CA2 (0.51) PTGS2CA2CA9CA1CA12
SCHEMBL31235134 0.80 CA2 (0.51) PTGS2CA2CA9CA1CA12
SCHEMBL30610973 0.79 HDAC3 (0.51) HDAC3HDAC1HDAC8ESR1ESR2
SCHEMBL28877972 0.76 PTGS2 (0.47) PTGS2CA2CA9CA1CA12
SCHEMBL28113571 0.76 HDAC3 (0.49) HDAC3HDAC1HDAC8ESR1ESR2
SCHEMBL29892589 0.75 KEAP1 (0.44) CA2CA9CA1CA12KDM4E
SCHEMBL28767740 0.75 CA2 (0.50) PTGS2CA2CA9CA1CA12
SCHEMBL29496941 0.74 SLC40A1 (0.42) CA2CA9CA1CA12MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2019238067-A1 PYRROLO [2, 3-B] PYRIDINES OR PYRROLO [2, 3-B] PYRAZINES AS HPK1 INHIBITOR AND THE USE THEREOF BEIGENE, LTD. (KY) 2019-12-19 WO disclosed