SCHEMBL21591735

SCHEMBL21591735

CCOC=Cc1cnc(OC)cc1CCNC(=O)O

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 13/20 0.45
MTNR1A P48039 12/20 0.45
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
NAMPT P43490 2/20 0.34
NNMT P40261 1/20 0.34
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21591699 0.76 MTNR1B (0.51) MTNR1BMTNR1ANNMT
SCHEMBL21591748 0.75 MTNR1B (0.50) MTNR1BMTNR1ANNMT
SCHEMBL23555513 0.75 L3MBTL1 (0.39) NNMT
SCHEMBL21591711 0.75 MTNR1A (0.53) MTNR1BMTNR1ANNMT
SCHEMBL23555514 0.74 NNMT (0.50) NNMT
SCHEMBL31088740 0.72 TUBB4A (0.33)
SCHEMBL31089176 0.71 TUBB4A (0.31)
SCHEMBL31089280 0.69 MAPT (0.40)
SCHEMBL31089007 0.68 ACVR2A (0.33)
SCHEMBL4315975 0.65 RECQL (0.43) MTNR1BMTNR1ANNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3807270-A1 NOVEL HETEROARYL HETEROCYCLYL COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. Hoffmann-La Roche AG (CH) 2021-04-21 EP disclosed
WO-2019238616-A1 NOVEL HETEROARYL HETEROCYCLYL COMPOUNDS FOR THE TREATMENT OF AUTOIMMUNE DISEASE F. HOFFMANN-LA ROCHE AG (CH) 2019-12-19 WO disclosed