Duvoglustat

Duvoglustat

SCHEMBL2163281

OCC1NCC(O)C(O)C1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GAAGLA

The experimentally established mechanism targets of Duvoglustat. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA known ✓ P10253 6/20 1.00
GLA known ✓ P06280 4/20 1.00
FUCA1 P04066 4/20 1.00
MGAM O43451 4/20 1.00
GBA2 Q9HCG7 3/20 1.00
SI P14410 3/20 1.00
AGL P35573 3/20 1.00
MEN1 O00255 2/20 1.00
ALOX15 P16050 2/20 1.00
KMT2A Q03164 2/20 1.00
GBA1 P04062 2/20 1.00
LCT P09848 2/20 1.00
GBA3 Q9H227 2/20 1.00
MAN2B1 O00754 1/20 1.00
MAN2B2 Q9Y2E5 1/20 1.00
ALDH1A1 P00352 1/20 1.00
CYP2C19 P33261 1/20 1.00
TREH O43280 1/20 1.00
GANAB Q14697 1/20 1.00
MGAM2 Q2M2H8 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Duvoglustat SCHEMBL13298786 1.00 GAA (1.00) GAAFUCA1GLAMGAMGBA2
Duvoglustat SCHEMBL4619759 1.00 GAA (1.00) GAAFUCA1GLAMGAMGBA2
Duvoglustat SCHEMBL15896653 1.00 GAA (1.00) GAAFUCA1GLAMGAMGBA2
Duvoglustat SCHEMBL142573 1.00 GAA (1.00) GAAFUCA1GLAMGAMGBA2
Duvoglustat SCHEMBL10028910 1.00 GAA (1.00) GAAFUCA1GLAMGAMGBA2
Duvoglustat SCHEMBL12269503 1.00 GAA (1.00) GAAFUCA1GLAMGAMGBA2
Duvoglustat SCHEMBL24518227 1.00 GAA (1.00) GAAFUCA1GLAMGAMGBA2
Duvoglustat SCHEMBL13061461 1.00 GAA (1.00) GAAFUCA1GLAMGAMGBA2
Duvoglustat SCHEMBL21104989 1.00 GAA (1.00) GAAFUCA1GLAMGAMGBA2
Duvoglustat SCHEMBL9015606 1.00 GAA (1.00) GAAFUCA1GLAMGAMGBA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 325 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115867534-A Non-lysosomal glucosylceramidase inhibitors and uses thereof 阿勒克图治疗公司 2023-03-28 CN claimed
CN-115010915-A Nitrogen branched nine-arm polyethylene glycol derivative, preparation method and biological related substance modified by nitrogen branched nine-arm polyethylene glycol derivative 厦门赛诺邦格生物科技股份有限公司 2022-09-06 CN claimed
US-11407768-B2 AMPK activators KALLYOPE, INC. (US) 2022-08-09 US claimed
US-11324827-B2 Multifunctionalized polyethylene glycol derivative and preparation method therefor XIAMEN SINOPEG BIOTECH CO., LTD. (CN) 2022-05-10 US claimed
CN-110643032-B Eight-arm polyethylene glycol, preparation method, functionalized derivative and modified biologically-relevant substance 厦门赛诺邦格生物科技股份有限公司 2022-01-28 CN claimed
CN-112694608-A Six-arm polyethylene glycol derivative, preparation method and modified biologically-relevant substance 厦门赛诺邦格生物科技股份有限公司 2021-04-23 CN claimed
CN-110643032-A Eight-arm polyethylene glycol, preparation method, functionalized derivative and modified biologically-relevant substance 厦门赛诺邦格生物科技股份有限公司 2020-01-03 CN claimed
CN-106967213-B Eight-arm polyethylene glycol, preparation method, functionalized derivative and modified biologically-relevant substance 厦门赛诺邦格生物科技股份有限公司 2019-11-05 CN claimed
EP-3315531-A1 8-ARM POLYETHYLENE GLYCOL DERIVATIVE, MANUFACTURING METHOD AND MODIFIED BIO-RELATED SUBSTANCE THEREBY Xiamen Sinopeg Biotech Co., Ltd. (CN) 2018-05-02 EP claimed
CN-104877127-B A kind of eight arms polyethyleneglycol derivative, preparation method and its bio-related substance of modification 厦门赛诺邦格生物科技股份有限公司 2017-11-10 CN claimed
US-20010049443-A1 Process for the preparation of 1,5-dideoxy-1,5-imino hexitols from oximes or imines BOARD OF TRUSTEES OPERATING MICHIGAN STATE UNIVERSITY (US) 2001-12-06 US claimed
WO-2001074776-A1 PROCESS FOR THE PREPARATION OF 1,5-DIDEOXY-1,5-IMINO HEXITOLS FROM OXIMES OR IMINES MICHIGAN STATE UNIVERSITY (US) 2001-10-11 WO claimed
US-5763438-A ANTIVIRAL AGENTS SEIKAGAKU CORPORATION (JP) 1998-06-09 US claimed
EP-0765865-A1 2-ACYLAMINOPROPANOL COMPOUND AND MEDICINAL COMPOSITION SEIKAGAKU CORPORATION (JP) 1997-04-02 EP claimed
US-4339585-A Method for the production of 2-hydroxymethyl-3,4,5-trihydroxy piperidine and the corresponding N-methyl derivative NIPPON SHINYAKU CO., LTD. (JP) 1982-07-13 US claimed
US-RE30886-E AND INHIBITING LIPID SYNTHESIS, USING 2-HYDROXYMETHYL-3,4,5-TRIHYDROXY-PIPERIDINE NIPPON SHINYAKU COMPANY LTD. (JP) 1982-03-23 US claimed
US-4312872-A TREATMENT OF ADIPOSITY, DIABETES, AND HYPERLIPOPROTEINEMIA BAYER AKTIENGESELLSCHAFT (DE) 1982-01-26 US claimed
US-4198481-A CULTURING STRAIN OF STREPTOMYCES NIPPON SHINYAKU CO., LTD. (JP) 1980-04-15 US claimed
US-4137231-A Process for the isolation of 2-hydroxymethyl-3,4,5-trihydroxypiperidine from plant material NIPPON SHINYAKU CO., LTD. (JP) 1979-01-30 US claimed
US-4065562-A 2-HYDROXYMETHYL-3,4,5-TRIHYDROXY-PIPERIDINE NIPPON SHINYAKU CO., LTD. (JA) 1977-12-27 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010049443-A1 Process for the preparation of 1,5-dideoxy-1,5-imino hexitols from oximes or imines GALE, HK1, G6PD GAA 914/4885GLA 349/4885FUCA1 1053/4885
US-11407768-B2 AMPK activators PRKAG1, PRKAG2, PRKAA1 GAA 784/4885GLA 1300/4885FUCA1 974/4885
US-11324827-B2 Multifunctionalized polyethylene glycol derivative and preparation method therefor HDGF, F11, F12 GAA 1797/4885GLA 1838/4885FUCA1 851/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.