SCHEMBL2170146

SCHEMBL2170146

COCCN1CCN(CC(=O)NC(Cc2ccc(Oc3ccc(F)cc3)cc2)C(N)=O)CC1

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 8/20 0.48
ALDH1A1 P00352 3/20 0.44
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
KMT2A Q03164 2/20 0.40
LMNA P02545 1/20 0.40
MEN1 O00255 1/20 0.40
TACR2 P21452 1/20 0.40
CNR2 P34972 1/20 0.40
STAT3 P40763 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2356486 0.91 SCN9A (0.45) SCN9AALDH1A1ITGB3ITGA2BTACR2
SCHEMBL2171096 0.87 SCN9A (0.51) SCN9AALDH1A1KMT2AMEN1
SCHEMBL2169958 0.86 SCN9A (0.47) SCN9AALDH1A1KMT2ALMNAMEN1
SCHEMBL2170108 0.85 LMNA (0.52) SCN9AALDH1A1KMT2ALMNAMEN1
SCHEMBL2171705 0.85 MEN1 (0.60) ALDH1A1KMT2ALMNAMEN1
SCHEMBL2170398 0.84 ALDH1A1 (0.51) SCN9AALDH1A1CNR2
SCHEMBL2171851 0.84 KMT2A (0.53) SCN9AALDH1A1KMT2ATACR2
SCHEMBL2169808 0.84 SCN9A (0.48) SCN9AALDH1A1TACR2
SCHEMBL2171621 0.84 QRFPR (0.50) SCN9AALDH1A1ITGB3ITGA2B
SCHEMBL2170811 0.83 MAPT (0.54) SCN9AALDH1A1KMT2ALMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed