SCHEMBL2170108

SCHEMBL2170108

NC(=O)C(Cc1ccc(Oc2ccc(F)cc2)cc1)NC(=O)CN1CCN(c2ccc(F)cc2)CC1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 5/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
ALDH1A1 P00352 2/20 0.52
REV1 Q9UBZ9 2/20 0.50
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
CA7 P43166 1/20 0.49
CA9 Q16790 1/20 0.49
DRD4 P21917 1/20 0.48
ALOX15 P16050 1/20 0.48
SCN9A Q15858 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
HTT P42858 2/20 0.48
MAPT P10636 3/20 0.47
POLB P06746 1/20 0.47
PARP1 P09874 1/20 0.46
PARP14 Q460N5 1/20 0.46
PARP10 Q53GL7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171705 0.95 MEN1 (0.60) LMNAMEN1KMT2AALDH1A1REV1
SCHEMBL2170811 0.95 MAPT (0.54) LMNAMEN1KMT2AALDH1A1REV1
SCHEMBL2171096 0.89 SCN9A (0.51) MEN1KMT2AALDH1A1SCN9APOLB
SCHEMBL2171851 0.89 KMT2A (0.53) KMT2AALDH1A1ALOX15SCN9A
SCHEMBL2170332 0.88 ALDH1A1 (0.53) LMNAMEN1KMT2AALDH1A1SCN9A
SCHEMBL2354704 0.88 ALDH1A1 (0.50) ALDH1A1CA1CA2CA7CA9
SCHEMBL2169958 0.87 SCN9A (0.47) LMNAMEN1KMT2AALDH1A1CA1
SCHEMBL2171621 0.87 QRFPR (0.50) ALDH1A1SCN9A
SCHEMBL2169808 0.87 SCN9A (0.48) ALDH1A1SCN9A
SCHEMBL2170146 0.85 SCN9A (0.48) LMNAMEN1KMT2AALDH1A1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed