SCHEMBL2170633

SCHEMBL2170633

CC(C(N)=O)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.67
PARP10 Q53GL7 1/20 0.60
LTA4H P09960 1/20 0.57
MAOB P27338 1/20 0.56
NPC1 O15118 1/20 0.55
RAB9A P51151 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
NR4A1 P22736 1/20 0.55
NR4A2 P43354 1/20 0.55
NR4A3 Q92570 1/20 0.55
RXRA P19793 1/20 0.55
RXRB P28702 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8833698 0.88 ALOX5 (0.62) ALOX5LTA4HMAOBNR4A1NR4A2
SCHEMBL2885897 0.88 ALOX5 (0.62) ALOX5LTA4HMAOBNR4A1NR4A2
Hydrochloric Acid SCHEMBL6948842 0.86 ALOX5 (0.60) ALOX5LTA4HMAOBNR4A1NR4A2
SCHEMBL6948837 0.85 ALOX5 (0.59) ALOX5LTA4HMAOBNR4A1NR4A2
SCHEMBL9577464 0.85 ALOX5 (0.59) ALOX5LTA4HMAOBNR4A1NR4A2
SCHEMBL28353364 0.84 MRGPRX4 (0.59) ALOX5PARP10MAOBNPC1RAB9A
SCHEMBL6266373 0.84 LTA4H (0.59) ALOX5LTA4HMAOBNPC1RAB9A
SCHEMBL7401422 0.82 LMNA (0.71) ALOX5MAOBNR4A1NR4A2NR4A3
SCHEMBL28724154 0.82 LMNA (0.70) ALOX5PARP10LTA4HMAOBNPC1
SCHEMBL28115187 0.82 PARP10 (0.60) ALOX5PARP10MAOBRAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349252-A2 SYNERGISTIC COMBINATION OF SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS AND ANTIMICROTUBULE AGENTS Exelixis, Inc. (US) 2011-08-03 EP disclosed
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed
EP-0337714-A2 HIV protease inhibitors useful for the treatment of aids MERCK & CO. INC. (US) 1989-10-18 EP disclosed