SCHEMBL6948837

SCHEMBL6948837

CC(C(=O)Cl)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.68

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.59
MAOB P27338 1/20 0.56
NR4A1 P22736 1/20 0.55
NR4A2 P43354 1/20 0.55
NR4A3 Q92570 1/20 0.55
RXRA P19793 1/20 0.55
RXRB P28702 1/20 0.55
LMNA P02545 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
FFAR1 O14842 1/20 0.54
ACACB O00763 1/20 0.54
LTA4H P09960 1/20 0.53
MRGPRX4 Q96LA9 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8833698 0.88 ALOX5 (0.62) ALOX5MAOBNR4A1NR4A2NR4A3
SCHEMBL2885897 0.88 ALOX5 (0.62) ALOX5MAOBNR4A1NR4A2NR4A3
Hydrochloric Acid SCHEMBL6948842 0.86 ALOX5 (0.60) ALOX5MAOBNR4A1NR4A2NR4A3
SCHEMBL2170633 0.85 ALOX5 (0.67) ALOX5MAOBNR4A1NR4A2NR4A3
SCHEMBL9577464 0.85 ALOX5 (0.59) ALOX5MAOBNR4A1NR4A2NR4A3
SCHEMBL6266373 0.84 LTA4H (0.59) ALOX5MAOBLMNAL3MBTL1ACACB
SCHEMBL28353364 0.84 MRGPRX4 (0.59) ALOX5MAOBNR4A1NR4A2NR4A3
SCHEMBL27733432 0.83 NR4A1 (0.57) ALOX5MAOBNR4A1NR4A2NR4A3
SCHEMBL7401422 0.82 LMNA (0.71) ALOX5MAOBNR4A1NR4A2NR4A3
SCHEMBL10867537 0.82 LMNA (0.70) ALOX5MAOBNR4A1NR4A2NR4A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3704117-B1 AZABICYCLO DERIVATIVES FOR TREATING OCULAR DISORDERS ALCON INC (CH) 2026-01-28 EP disclosed
US-12247028-B2 Azabicyclo and diazepine derivatives ALCON INC. (CH) 2025-03-11 US disclosed
US-20240132497-A1 AZABICYCLO AND DIAZEPINE DERIVATIVES ALCON INC. (CH) 2024-04-25 US disclosed
US-11884666-B2 Azabicyclo and diazepine derivatives ALCON INC. (CH) 2024-01-30 US disclosed
US-20220267328-A1 AZABICYCLO AND DIAZEPINE DERIVATIVES ALCON INC. (CH) 2022-08-25 US disclosed
US-11306090-B2 Azabicyclo and diazepine derivatives ALCON INC. (CH) 2022-04-19 US disclosed
US-20210179616-A1 AZABICYCLO AND DIAZEPINE DERIVATIVES ALCON INC. (CH) 2021-06-17 US disclosed
US-20210179616-A1 AZABICYCLO AND DIAZEPINE DERIVATIVES ALCON INC. (CH) 2021-06-17 US disclosed
EP-3704117-A1 AZABICYCLO AND DIAZEPINE DERIVATIVES FOR TREATING OCULAR DISORDERS ALCON INC. (CH) 2020-09-09 EP disclosed
CN-111247147-A Azabicyclo and diazepatriene derivatives useful for treating ocular disorders 爱尔康公司 2020-06-05 CN disclosed
EP-0936218-B1 BENZIMIDAZOLE DERIVATIVES MOCHIDA PHARM CO LTD (JP) 2003-04-02 EP disclosed
US-6387938-B1 Benzimidazole derivatives MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 2002-05-14 US disclosed
US-5952390-A ANTIINFLAMMATORY AGENTS; TREATMENT FOR PSORIASIS TEVA PHARMACEUTICAL INDUSTRIES LTD. (IL) 1999-09-14 US disclosed
EP-0936218-A1 NOVEL BENZIMIDAZOLE DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1999-08-18 EP disclosed
US-5844004-A 10-substituted 1,8-dihydroxy-9 (10H) anthracenone pharmaceuticals TEVA PHARMACEUTICAL INDUSTRIES, LTD. (IL) 1998-12-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11884666-B2 Azabicyclo and diazepine derivatives CHRM3, CHRM5, CHRNA5 ALOX5 867/4885MAOB 376/4885NR4A1 236/4885
US-20240132497-A1 AZABICYCLO AND DIAZEPINE DERIVATIVES CHRM3, CHRM5, CHRNA5 ALOX5 867/4885MAOB 376/4885NR4A1 236/4885
US-20210179616-A1 AZABICYCLO AND DIAZEPINE DERIVATIVES CHRM3, CHRM5, CHRNA5 ALOX5 867/4885MAOB 376/4885NR4A1 236/4885
US-20220267328-A1 AZABICYCLO AND DIAZEPINE DERIVATIVES CHRM3, CHRM5, CHRNA5 ALOX5 867/4885MAOB 376/4885NR4A1 236/4885
US-12247028-B2 Azabicyclo and diazepine derivatives CHRM3, CHRM5, CHRNA5 ALOX5 867/4885MAOB 376/4885NR4A1 236/4885
US-11306090-B2 Azabicyclo and diazepine derivatives CHRM3, CHRM5, CHRNA5 ALOX5 867/4885MAOB 376/4885NR4A1 236/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.