SCHEMBL21708795

SCHEMBL21708795

CCCC(F)OC(=O)CC(C)(C#N)c1ccccc1Cl

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 1/20 0.33
TAS1R1 Q7RTX1 1/20 0.33
CTSK P43235 1/20 0.30
ALDH1A1 P00352 1/20 0.30
CASP1 P29466 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708740 0.89 L3MBTL1 (0.32) TAS1R3TAS1R1ALDH1A1
SCHEMBL21708706 0.87 L3MBTL1 (0.32) TAS1R3TAS1R1CTSKALDH1A1
SCHEMBL21708670 0.86 MEN1 (0.36) TAS1R3TAS1R1CTSKALDH1A1
SCHEMBL21708771 0.84 SMN1; SMN2 (0.34) ALDH1A1
SCHEMBL21708759 0.83 NPC1 (0.32) TAS1R3TAS1R1
SCHEMBL21708704 0.81 TAS1R3 (0.33) TAS1R3TAS1R1CTSKALDH1A1
SCHEMBL21656302 0.78 CTSS (0.34) CTSKALDH1A1
SCHEMBL21708649 0.77 NR3C1 (0.39) TAS1R3TAS1R1
SCHEMBL21708724 0.76 NR3C2 (0.35) TAS1R3TAS1R1
SCHEMBL21631919 0.75 CYP2C19 (0.42) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed