SCHEMBL21708683

SCHEMBL21708683

CCCC(F)OC(=O)CC(CN)c1cccc(C)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
F10 P00742 8/20 0.38
F2 P00734 7/20 0.38
PRSS1 P07477 5/20 0.38
GABBR2 O75899 1/20 0.38
GABBR1 Q9UBS5 1/20 0.38
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
ROCK2 O75116 1/20 0.35
GAA P10253 1/20 0.34
PSEN1 P49768 1/20 0.34
PSEN2 P49810 1/20 0.34
APH1B Q8WW43 1/20 0.34
NCSTN Q92542 1/20 0.34
APH1A Q96BI3 1/20 0.34
PSENEN Q9NZ42 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
SLC6A3 Q01959 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708787 0.87 HPGD (0.39) F10F2PRSS1GABBR2GABBR1
SCHEMBL21708681 0.86 L3MBTL1 (0.46) TAS1R3TAS1R1ROCK2GAA
SCHEMBL21708638 0.85 GABBR2 (0.38) F10F2GABBR2GABBR1GAA
SCHEMBL21708758 0.81 ROCK2 (0.45) TAS1R3TAS1R1ROCK2PSEN1PSEN2
SCHEMBL21708755 0.80 KMT2A (0.38) TAS1R3TAS1R1GAAPSEN1PSEN2
SCHEMBL21708766 0.78 GABBR2 (0.33) F10F2GABBR2GABBR1ROCK2
SCHEMBL21708792 0.78 TAS1R3 (0.33) F10F2PRSS1GABBR2GABBR1
SCHEMBL21656318 0.76 GABBR2 (0.42) F10F2PRSS1GABBR2GABBR1
SCHEMBL23750383 0.75 GABBR2 (0.49) GABBR2GABBR1ROCK2GAACYP1A2
SCHEMBL23750224 0.75 GABBR2 (0.49) GABBR2GABBR1ROCK2GAACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed