SCHEMBL21708759

SCHEMBL21708759

CCCC(F)OC(=O)CC(C)(C#N)c1ncccc1Cl

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
GAA P10253 2/20 0.31
ANO1 Q5XXA6 1/20 0.31
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
BDKRB1 P46663 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
PLCG1 P19174 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708765 0.83 PLCG1 (0.33) NPC1RAB9AGAAANO1MEN1
SCHEMBL21708795 0.83 TAS1R3 (0.33) TAS1R3TAS1R1
SCHEMBL21708790 0.82 NPC1 (0.32) NPC1RAB9AANO1KMT2A
SCHEMBL21708771 0.80 SMN1; SMN2 (0.34) MEN1KMT2ASMN1; SMN2
SCHEMBL21656332 0.80 POLB (0.36) NPC1RAB9AGAABDKRB1SMN1; SMN2
SCHEMBL21631952 0.77 PTGFR (0.39) BDKRB1SMN1; SMN2PLCG1
SCHEMBL21708779 0.75 NPC1 (0.33) NPC1RAB9AGAAANO1TAS1R3
SCHEMBL21708740 0.74 L3MBTL1 (0.32) TAS1R3TAS1R1
SCHEMBL21708670 0.74 MEN1 (0.36) NPC1RAB9AGAATAS1R3TAS1R1
SCHEMBL21708706 0.73 L3MBTL1 (0.32) TAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed