SCHEMBL21708765

SCHEMBL21708765

CCCC(F)OC(=O)C(C)(C#N)c1ncccc1Cl

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLCG1 P19174 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
ANO1 Q5XXA6 1/20 0.32
KMT2A Q03164 2/20 0.31
MEN1 O00255 1/20 0.31
GAA P10253 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
ALDH1A1 P00352 2/20 0.30
ATM Q13315 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
USP9X Q93008 1/20 0.30
KDM4E B2RXH2 1/20 0.30
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30
PRSS1 P07477 1/20 0.30
CTSG P08311 1/20 0.30
CTRB1 P17538 1/20 0.30
CMA1 P23946 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708759 0.83 NPC1 (0.32) PLCG1NPC1RAB9AANO1KMT2A
SCHEMBL21708779 0.81 NPC1 (0.33) NPC1RAB9AANO1KMT2AGAA
SCHEMBL21708691 0.79 LMNA (0.36) RAB9AKMT2AGAASMN1; SMN2ALDH1A1
SCHEMBL21656559 0.78 PLCG1 (0.39) PLCG1SMN1; SMN2TDP1KDM4EPRSS1
SCHEMBL21708790 0.75 NPC1 (0.32) NPC1RAB9AANO1KMT2AALDH1A1
SCHEMBL21708674 0.75 ADRB2 (0.33) KMT2AMEN1L3MBTL1PRSS1CTSG
SCHEMBL21631946 0.74 SLC22A12 (0.38) PLCG1KMT2AMEN1GAASMN1; SMN2
SCHEMBL21708762 0.72 KMT2A (0.37) NPC1RAB9AKMT2AMEN1GAA
SCHEMBL21708795 0.69 TAS1R3 (0.33) ALDH1A1
SCHEMBL31368866 0.67 KMT2A (0.33) NPC1RAB9AKMT2AGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3609869-A1 SUBSTITUTED N-ARYLETHYL-2-ARYLQUINOLINE-4-CARBOXAMIDES AND USE THEREOF Bayer Aktiengesellschaft (DE) 2020-02-19 EP disclosed