SCHEMBL21709149

SCHEMBL21709149

C#CCOC(CN)c1cc(O)c(O)cc1C#C

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ADRB2 P07550 1/20 0.33
CYP3A4 P08684 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
ADRA1A P35348 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 1/20 0.33
APEX1 P27695 1/20 0.33
RAD52 P43351 1/20 0.33
RECQL P46063 1/20 0.33
BLM P54132 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
P2RX3 P56373 1/20 0.32
P2RX2 Q9UBL9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21709245 0.88 P2RX3 (0.31) P2RX3P2RX2
SCHEMBL21709247 0.81 LOXL2 (0.32) P2RX3P2RX2
SCHEMBL21709143 0.80
SCHEMBL21709151 0.80 MAOA (0.32)
SCHEMBL21709270 0.79 P2RX3 (0.38) ADRA2AADRA1AP2RX3P2RX2
SCHEMBL21708883 0.77
SCHEMBL21709162 0.75 TSHR (0.33)
SCHEMBL21708869 0.74 TDP1 (0.49) ADRB2CYP3A4HSD17B10ADRA2AADRA2B
SCHEMBL21708902 0.71 ADRA2A (0.35) ADRB2CYP3A4HSD17B10ADRA2AADRA2B
SCHEMBL21709214 0.71

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020032080-A1 COMPOUND, SALT OF COMPOUND, NEUROMODULATION AGENT, METHOD FOR EVALUATING NEUROMODULATION AGENT, METHOD FOR PRODUCING COMPOUND, AND METHOD FOR PRODUCING SALT OF COMPOUND 学校法人慶應義塾 2020-02-13 WO disclosed