SCHEMBL21728869

SCHEMBL21728869

NC(=O)Cc1cccc(CC(=O)O)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.58
CYP1A2 P05177 1/20 0.53
CYP2C19 P33261 1/20 0.53
LMNA P02545 2/20 0.48
GAA P10253 2/20 0.48
TSHR P16473 2/20 0.48
KDM4E B2RXH2 1/20 0.48
RGS12 O14924 1/20 0.48
POLB P06746 1/20 0.48
MAPT P10636 1/20 0.48
HPGD P15428 1/20 0.48
NFKB1 P19838 1/20 0.48
APEX1 P27695 1/20 0.48
THPO P40225 1/20 0.48
BLM P54132 1/20 0.48
GNAI1 P63096 1/20 0.48
PMP22 Q01453 1/20 0.48
HIF1A Q16665 1/20 0.48
HSD17B10 Q99714 1/20 0.48
TDP1 Q9NUW8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10339219 0.91 CA2 (0.54) LMNAKDM4EPOLBHPGDNFKB1
SCHEMBL70565 0.89 AKR1B1 (0.71) AKR1B1CYP1A2CYP2C19LMNAGAA
Hydrochloric Acid SCHEMBL8922940 0.87 AKR1B1 (0.68) AKR1B1CYP1A2CYP2C19LMNAGAA
SCHEMBL20634078 0.87 CA2 (0.48) AKR1B1LMNAGAATSHRKDM4E
SCHEMBL27697776 0.85 KEAP1 (0.57) PLA2G10PLA2G2AITGB3ITGA2B
SCHEMBL7557354 0.84 PLA2G2A (0.53) LMNAKDM4EHPGDNFKB1PLA2G10
SCHEMBL3803115 0.83 AKR1B1 (0.58) AKR1B1CYP1A2CYP2C19LMNAGAA
SCHEMBL31346922 0.83 PRSS1 (0.50) LMNATSHRKDM4EPOLBCA2
SCHEMBL28031264 0.83 PRSS1 (0.50) LMNATSHRKDM4EPOLBCA2
SCHEMBL7770968 0.83 ENPP2 (0.52) KDM4ENFKB1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3186270-B1 CYCLIC UREA COMPOUNDS AS GRANZYME B INHIBITORS VIDA THERAPEUTICS INC (CA) 2020-02-19 EP disclosed