SCHEMBL21733378

SCHEMBL21733378

COC[C@@H]1CC(F)CN1C

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 0.36
CASP7 P55210 4/20 0.36
NOS1 P29475 1/20 0.31
PDK1 Q15118 2/20 0.30
PDK2 Q15119 1/20 0.30
PDK3 Q15120 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10273862 1.00 CASP3 (0.36) CASP3CASP7NOS1PDK1PDK2
SCHEMBL21733403 1.00 CASP3 (0.36) CASP3CASP7NOS1PDK1PDK2
SCHEMBL23957329 1.00 CASP3 (0.36) CASP3CASP7NOS1PDK1PDK2
SCHEMBL24176145 1.00 CASP3 (0.36) CASP3CASP7NOS1PDK1PDK2
SCHEMBL18461688 0.85 ALOX5 (0.33)
SCHEMBL23158043 0.82 NOS1 (0.30) NOS1
SCHEMBL23158046 0.82 NOS1 (0.30) NOS1
SCHEMBL22062833 0.80
SCHEMBL24854605 0.80 PDK1 (0.33) PDK1
SCHEMBL22062975 0.79 ALDH1A1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4223761-A1 QUINAZOLINE COMPOUND AND APPLICATION THEREOF Shanghai Pharmaceuticals Holding Co., Ltd. (CN) 2023-08-09 EP disclosed
WO-2023125627-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND AND APPLICATION THEREOF LYNK PHARMACEUTICALS CO., LTD. (CN) 2023-07-06 WO disclosed
WO-2023086383-A1 SELECT KRAS G12C INHIBITORS AND USES THEREOF 1200 PHARMA LLC (US) 2023-05-19 WO disclosed
WO-2022262797-A1 COMBINATION OF AN ERK INHIBITOR AND A KRAS INHIBITOR AND USES THEREOF SHANGHAI ANTENGENE CORPORATION LIMITED (CN) 2022-12-22 WO disclosed
WO-2022266015-A1 FUSED HETEROARYL COMPOUNDS USEFUL AS ANTICANCER AGENTS KUMQUAT BIOSCIENCES INC. (US) 2022-12-22 WO disclosed
WO-2020035031-A1 FUSED RING COMPOUNDS GENENTECH, INC. (US) 2020-02-20 WO disclosed