SCHEMBL2173714

SCHEMBL2173714

NC(=O)C(Cc1ccc(Oc2ccc(F)cc2)cc1)NC(=O)CN1CCC(N2CCCC2)CC1

nearest known ligand 0.45

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 5/20 0.45
HPGD P15428 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
HRH3 Q9Y5N1 9/20 0.40
ALDH1A1 P00352 2/20 0.39
PARP1 P09874 2/20 0.39
KCNH2 Q12809 1/20 0.39
KDM4E B2RXH2 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2171096 0.90 SCN9A (0.51) SCN9AHPGDMEN1KMT2AALDH1A1
SCHEMBL2170398 0.87 ALDH1A1 (0.51) SCN9AALDH1A1KDM4E
SCHEMBL2185323 0.84 SCN9A (0.45) SCN9AHPGDMEN1KMT2A
SCHEMBL2171621 0.83 QRFPR (0.50) SCN9AALDH1A1
SCHEMBL2169808 0.83 SCN9A (0.48) SCN9AALDH1A1
SCHEMBL2171851 0.83 KMT2A (0.53) SCN9AHPGDKMT2AALDH1A1
SCHEMBL2170108 0.82 LMNA (0.52) SCN9AMEN1KMT2AALDH1A1PARP1
SCHEMBL2350905 0.82 HPGD (0.48) SCN9AHPGDMEN1KMT2AHRH3
SCHEMBL2169958 0.82 SCN9A (0.47) SCN9AMEN1KMT2AHRH3ALDH1A1
SCHEMBL2170146 0.80 SCN9A (0.48) SCN9AMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed