SCHEMBL21759880

SCHEMBL21759880

CC/C=C\c1ncccc1CC

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.35
ALDH1A1 P00352 2/20 0.35
GABRA1 P14867 2/20 0.34
GABRB2 P47870 2/20 0.34
HTR1A P08908 1/20 0.34
TAAR1 Q96RJ0 1/20 0.34
NFE2L2 Q16236 7/20 0.33
CYP1A2 P05177 1/20 0.33
MAPT P10636 1/20 0.33
LMNA P02545 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
HPGD P15428 1/20 0.32
HSD17B10 Q99714 1/20 0.32
SGMS2 Q8NHU3 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9000359 0.85 SLC40A1 (0.37) KDM4EALDH1A1GABRA1GABRB2HTR1A
SCHEMBL11830127 0.85 KDM4E (0.35) KDM4EALDH1A1GABRA1GABRB2HTR1A
SCHEMBL6115316 0.80 TRIM24 (0.39) KDM4EALDH1A1GABRA1GABRB2HTR1A
SCHEMBL659486 0.80 GABRA1 (0.37) KDM4EALDH1A1GABRA1GABRB2HTR1A
SCHEMBL472968 0.78 LMNA (0.37) KDM4EALDH1A1GABRA1GABRB2HTR1A
SCHEMBL22239425 0.78 NOS3 (0.42) KDM4ECYP1A2MAPTLMNAL3MBTL1
Benzene SCHEMBL11824212 0.77 TRIM24 (0.37) KDM4EALDH1A1GABRA1GABRB2HTR1A
SCHEMBL18215495 0.77 NFE2L2 (0.51) NFE2L2
SCHEMBL18024029 0.77 RRM1 (0.41) KDM4EALDH1A1CYP1A2MAPTLMNA
SCHEMBL18802147 0.76 GRIN1 (0.35) KDM4EALDH1A1GABRA1GABRB2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2585462-B1 FUSED HETEROCYCLIC COMPOUNDS AS PHOSPHODIESTERASES (PDES) INHIBITORS TAKEDA PHARMACEUTICALS CO (JP) 2020-02-26 EP disclosed