SCHEMBL21789030

SCHEMBL21789030

CC(C)(C)[Si](C)(C)OCC12CC(C1)[C@@H](C(=O)c1ccccc1)C2

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 1/20 0.34
TOP2A P11388 1/20 0.33
AVPR1A P37288 3/20 0.33
EHMT2 Q96KQ7 2/20 0.32
CYP3A4 P08684 3/20 0.32
SRC P12931 1/20 0.32
CES1 P23141 1/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
KMT2A Q03164 1/20 0.31
P2RX7 Q99572 1/20 0.31
GAA P10253 1/20 0.31
BACE1 P56817 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21788901 0.74 LMNA (0.42) TOP2AAVPR1AEHMT2CYP3A4SRC
SCHEMBL21789249 0.73
SCHEMBL21777934 0.72 TSHR (0.38) AVPR1ACYP3A4MEN1ALDH1A1CYP1A2
SCHEMBL8447329 0.71 CHRNB2 (0.41) CYP3A4ALDH1A1GAA
SCHEMBL21788880 0.68 TOP2A (0.40) TOP2AAVPR1ACYP3A4ALDH1A1CYP1A2
SCHEMBL16148176 0.68 TSHR (0.38) TOP2AAVPR1ACYP3A4MEN1ALDH1A1
SCHEMBL1712501 0.67 NPC1 (0.45) CYP3A4CES1MEN1ALDH1A1CYP1A2
SCHEMBL24165052 0.65 ALDH1A1 (0.42) CYP3A4MEN1ALDH1A1CYP1A2CYP2C9
SCHEMBL9433444 0.65 L3MBTL1 (0.46) CYP3A4CES1MEN1ALDH1A1CYP1A2
SCHEMBL28498515 0.65 MAPK1 (0.50) ALDH1A1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020047447-A1 CARDIAC SARCOMERE INHIBITORS CYTOKINETICS, INC. (US) 2020-03-05 WO disclosed