SCHEMBL21795658

SCHEMBL21795658

NC(=O)O[C@H]1CCOC[C@@H]1COc1ccc(Cn2cccn2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
NOS3 P29474 1/20 0.38
NOS1 P29475 1/20 0.38
FFAR4 Q5NUL3 3/20 0.38
KLKB1 P03952 3/20 0.37
TDP1 Q9NUW8 1/20 0.37
HRH3 Q9Y5N1 3/20 0.37
GAA P10253 2/20 0.36
MAPT P10636 2/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA9 Q16790 1/20 0.36
MAOB P27338 1/20 0.35
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15420605 0.81 HDAC1 (0.41) HDAC1HDAC6FFAR4KLKB1TDP1
SCHEMBL15420406 0.77 CA12 (0.38) HDAC1HDAC6HRH3GAAMAPT
SCHEMBL21795640 0.75 PARP15 (0.42) HRH3GAAMAPTMAOBKDM4E
SCHEMBL21795659 0.75 NPC1 (0.39) FFAR4MAPTNPC1RAB9ASMN1; SMN2
SCHEMBL21795643 0.74 DDB1 (0.38) FFAR4NPC1RAB9AHTT
SCHEMBL21795648 0.73 XDH (0.39) FFAR4MAOB
SCHEMBL21795636 0.73 XDH (0.39) FFAR4MAOB
SCHEMBL21795642 0.72 GCG (0.34) HDAC1HDAC6FFAR4
SCHEMBL12989127 0.71 BCHE (0.45)
SCHEMBL12989126 0.71 BCHE (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2694472-B1 SULFONAMIDE DERIVATIVE AND USE THEREOF TAKEDA PHARMACEUTICALS CO (JP) 2020-03-11 EP disclosed